SCHEMBL12880591

SCHEMBL12880591

BrC(c1ccccc1)c1ccc(-c2ccc(C(Br)c3ccccc3)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.50
CHRNA4 P43681 1/20 0.50
ACP3 P15309 2/20 0.45
ALDH1A1 P00352 3/20 0.43
MAPK1 P28482 2/20 0.43
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
TRPA1 O75762 1/20 0.42
PTGS2 P35354 1/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
DPP4 P27487 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8721667 0.97 CHRNB2 (0.54) CHRNB2CHRNA4ACP3ALDH1A1MAPK1
SCHEMBL11218980 0.94 ALDH1A1 (0.50) CHRNB2CHRNA4ACP3ALDH1A1MAPK1
SCHEMBL12880577 0.91 CES2 (0.48) CHRNB2CHRNA4MAPK1CES2CES1
SCHEMBL67123 0.88 CES2 (0.50) MAPK1CES2CES1TRPA1CYP2D6
SCHEMBL11642941 0.84 CHRNB2 (0.42) CHRNB2CHRNA4ACP3ALDH1A1MAPK1
SCHEMBL11576225 0.81 HTR2A (0.58) ALDH1A1MAPK1CES2CES1TRPA1
SCHEMBL14528562 0.79 CES2 (0.39) CHRNB2CHRNA4CES2CES1TRPA1
SCHEMBL1528588 0.79 IDO1 (0.54) ALDH1A1MAPK1TRPA1CYP3A4CYP2D6
SCHEMBL7520122 0.79 LMNA (0.42) ALDH1A1CES2CES1TRPA1USP2
SCHEMBL1272990 0.79 LMNA (0.48) CES2CES1TRPA1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
EP-1623471-B1 METHOD FOR CONTROLLING THE MOLECULAR WEIGHT DURING POLY(ARYLENE VINYLENE) SYNTHESIS, AND POLYMERS PRODUCED THEREWITH MERCK PATENT GMBH (DE) 2007-05-30 EP disclosed