SCHEMBL12907214

SCHEMBL12907214

Cc1cn(-c2ccc(N3CCN(c4ccc(-c5ccccc5)cc4)CC3)cc2)cn1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP19A1 P11511 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CYP2E1 P05181 1/20 0.45
CYP2A6 P11509 1/20 0.45
DHFR P00374 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
NLRP3 Q96P20 1/20 0.44
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
TSHR P16473 2/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12907955 0.80 MAOA (0.40) MAOAMAOBCYP1A2CYP3A4CYP2D6
SCHEMBL2283022 0.80 CYP2E1 (0.65) MAOAMAOBCYP1A2CYP3A4CYP2D6
SCHEMBL12906832 0.80 MAPT (0.65) CYP2C9MAPTMEN1KMT2AALDH1A1
SCHEMBL27985278 0.78 CYP1A2 (0.65) MAOAMAOBCYP1A2CYP3A4CYP2D6
SCHEMBL12906826 0.77 CYP2E1 (0.42) MAOAMAOBCYP1A2CYP3A4CYP2D6
SCHEMBL12907213 0.75 NR2E1 (0.45) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL12906757 0.75 L3MBTL1 (0.43) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL7607579 0.75 HTR7 (0.59) CYP1A2CYP2C9CYP2C19NPC1RAB9A
Fluoride SCHEMBL27569822 0.74 MEN1 (0.56) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL12906825 0.73 PSEN1 (0.40) MAOAMAOBCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011016559-A1 HETEROCYCLIC COMPOUND AND USE THEREOF 武田薬品工業株式会社 (JP) 2011-02-10 WO disclosed