SCHEMBL12933366

SCHEMBL12933366

COc1ccc(N(CC(C)(C)C)C(=O)Nc2ccc(Oc3ccccc3)cc2)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.48
NPY5R Q15761 3/20 0.47
PGR P06401 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HPGD P15428 1/20 0.46
LMNA P02545 2/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
ALOX12 P18054 1/20 0.46
RAB9A P51151 1/20 0.46
MTNR1B P49286 4/20 0.45
MTNR1A P48039 3/20 0.45
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HTT P42858 1/20 0.44
GAA P10253 1/20 0.44
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12933367 0.92 LMNA (0.47) SMN1; SMN2HPGDLMNAMEN1KMT2A
SCHEMBL8345899 0.88 MCHR1 (0.56) MCHR1NPY5RPGRSMN1; SMN2HPGD
SCHEMBL12933363 0.87 IMPDH2 (0.54) SMN1; SMN2MEN1KMT2ARAB9AMAPT
SCHEMBL12963481 0.86 MCHR1 (0.54) MCHR1NPY5RPGRSMN1; SMN2HPGD
SCHEMBL12933364 0.85 MEN1 (0.50) SMN1; SMN2MEN1KMT2ARAB9AMAPT
SCHEMBL8347783 0.79 MEN1 (0.65) MCHR1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL12963493 0.77 MEN1 (0.51) MCHR1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL13074283 0.76 QPCT (0.51) SMN1; SMN2LMNAMEN1KMT2ARAB9A
SCHEMBL1058480 0.75 HDAC1 (0.59) MCHR1
SCHEMBL8348684 0.75 MCHR1 (0.67) MCHR1SMN1; SMN2HPGDLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed
US-7838520-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2010-11-23 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed