SCHEMBL13069050

SCHEMBL13069050

CC=C/C=C\C1=C(C)NC(=O)C12Cc1ccc(Nc3cc(C(=O)N4CCc5ccccc54)ncn3)cc1C2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.34
ALDH1A1 P00352 6/20 0.34
LMNA P02545 2/20 0.34
GAA P10253 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
SMN1; SMN2 Q16637 6/20 0.34
POLB P06746 1/20 0.34
ALOX15 P16050 1/20 0.34
NR4A1 P22736 1/20 0.34
CRBN Q96SW2 2/20 0.34
RAB9A P51151 6/20 0.33
NPC1 O15118 4/20 0.33
MAPT P10636 3/20 0.33
PKM P14618 2/20 0.33
NFKB1 P19838 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13846777 0.96 ALDH1A1 (0.38) ALDH1A1LMNASMN1; SMN2CRBNRAB9A
SCHEMBL13068721 0.91 NAMPT (0.31) POLBALOX15NR4A1
SCHEMBL13069055 0.88 ALOX15 (0.37) SPRALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL13068974 0.87 CALCRL (0.33) ALDH1A1SMN1; SMN2KDM4EMAPK1TP53
SCHEMBL13068645 0.85 GRM5 (0.35) ALDH1A1POLBKDM4EHPGDCALCRL
SCHEMBL13068728 0.85 GRM5 (0.35) ALDH1A1POLBKDM4EHPGDCALCRL
SCHEMBL13069029 0.85 EIF2AK3 (0.35)
SCHEMBL13846647 0.82
SCHEMBL13068671 0.81 GRM5 (0.36)
SCHEMBL13846735 0.81 MMP13 (0.41) ALDH1A1POLBMAPTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2251339-A2 COMPOUNDS Boehringer Ingelheim International GmbH (DE) 2010-11-17 EP disclosed
WO-2009065920-A2 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-05-28 WO disclosed