SCHEMBL13073299

SCHEMBL13073299

O=C1c2c(Cl)cccc2-n2ccnc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
IDO2 Q6ZQW0 1/20 0.46
NSD2 O96028 1/20 0.37
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRA5 P31644 3/20 0.36
HCAR1 Q9BXC0 4/20 0.36
GABRA1 P14867 2/20 0.35
GABRA3 P34903 2/20 0.35
GABRA2 P47869 2/20 0.35
GABRA6 Q16445 2/20 0.35
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRB1 P18505 1/20 0.34
GRM5 P41594 1/20 0.34
GABRB2 P47870 1/20 0.34
GABRA4 P48169 1/20 0.34
GABRE P78334 1/20 0.34
GABRG1 Q8N1C3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24857937 0.81 HCAR1 (0.33) GABRG2GABRB3GABRA5HCAR1GABRA1
SCHEMBL4730158 0.73 IDO1 (0.45) IDO1TDO2IDO2NSD2CES1
SCHEMBL15144565 0.69 HCAR1 (0.49) HCAR1
SCHEMBL27987583 0.68 IDO1 (0.49) IDO1TDO2IDO2GABRG2GABRB3
SCHEMBL27987592 0.68 IDO1 (0.45) IDO1TDO2IDO2HCAR1CES1
SCHEMBL8558631 0.67 HSD11B1 (0.58) HCAR1MET
SCHEMBL9885126 0.67 IDO1 (0.68) IDO1TDO2IDO2
SCHEMBL27522182 0.67 LMNA (0.40) GABRG2GABRB3GABRA5
SCHEMBL28923906 0.66 P2RX7 (0.43) HCAR1
SCHEMBL12342913 0.66 CYP3A4 (0.47) HCAR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010132352-A2 SPIRO COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2010-11-18 WO disclosed