SCHEMBL13087758

SCHEMBL13087758

COC(=O)c1cccc(Oc2ccc(C(=O)O)cc2)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.65
SRD5A2 P31213 2/20 0.56
TNKS O95271 1/20 0.55
PARP15 Q460N3 1/20 0.55
PARP14 Q460N5 1/20 0.55
PARP10 Q53GL7 1/20 0.55
TNKS2 Q9H2K2 1/20 0.55
PARP2 Q9UGN5 1/20 0.55
KMO O15229 1/20 0.55
KDM4E B2RXH2 1/20 0.55
NPC1 O15118 2/20 0.55
POLB P06746 2/20 0.55
RAB9A P51151 2/20 0.55
CYP2C9 P11712 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
ALDH1A1 P00352 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
NR1H4 Q96RI1 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.51
PGR P06401 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31657173 0.94 AKR1C3 (0.70) AKR1C3TNKSPARP15PARP14PARP10
SCHEMBL883130 0.92 TNKS (0.60) AKR1C3TNKSPARP15PARP14PARP10
SCHEMBL521860 0.90 AKR1C3 (0.68) AKR1C3TNKSPARP15PARP14PARP10
SCHEMBL2436534 0.88 L3MBTL1 (0.65) AKR1C3TNKSPARP15PARP14PARP10
SCHEMBL70012 0.87 AKR1C3 (0.85) AKR1C3SRD5A2TNKSPARP15PARP14
SCHEMBL30307447 0.87 AKR1C3 (0.85) AKR1C3SRD5A2TNKSPARP15PARP14
SCHEMBL16429240 0.87 AKR1C3 (0.85) AKR1C3SRD5A2TNKSPARP15PARP14
SCHEMBL28051885 0.86 AKR1C3 (0.67) AKR1C3SRD5A2TNKSPARP15PARP14
SCHEMBL14217726 0.86 L3MBTL1 (0.56) AKR1C3TNKSPARP15PARP14PARP10
Hydrochloric Acid SCHEMBL7137782 0.85 AKR1C3 (0.82) AKR1C3SRD5A2TNKSPARP15PARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020009156-A1 BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVE 第一三共株式会社 2020-01-09 WO disclosed
WO-2010117635-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-10-14 WO disclosed