SCHEMBL13102415

SCHEMBL13102415

CC(C)Cc1nc2cccc(F)c2c(=O)n1NC(=O)Cc1cccc(OC(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 1/20 0.41
FFAR2 O15552 1/20 0.40
GLS O94925 8/20 0.40
GPR139 Q6DWJ6 2/20 0.40
CSNK1D P48730 1/20 0.39
RORC P51449 1/20 0.39
CTSD P07339 1/20 0.39
RIPK1 Q13546 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13102403 0.91 TRPV4 (0.43) P2RY14GPR139
SCHEMBL13101690 0.88 ALDH1A1 (0.49) P2RY14GPR139
SCHEMBL13102005 0.87 KDM4E (0.43) FFAR2GPR139CSNK1DRIPK1
SCHEMBL13102401 0.87 GLS (0.39) FFAR2GLS
SCHEMBL13102078 0.86 SLC2A1 (0.43) P2RY14FFAR2GLSGPR139CSNK1D
SCHEMBL13101980 0.86 GPR139 (0.46) P2RY14FFAR2GPR139CSNK1DCTSD
SCHEMBL13102285 0.86 NPSR1 (0.44)
SCHEMBL13102493 0.85 ALDH1A1 (0.40) GPR139
SCHEMBL13102419 0.84 MEN1 (0.39) GPR139
SCHEMBL13101991 0.83 RORC (0.41) P2RY14GPR139RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329713-B2 Fused ring heterocycles as potassium channel modulators ICAGEN INC. (US) 2012-12-11 US disclosed
US-20100273784-A1 FUSED RING HETEROCYCLES AS POTASSIUM CHANNEL MODULATORS ICAGEN, INC. (US) 2010-10-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100273784-A1 FUSED RING HETEROCYCLES AS POTASSIUM CHANNEL MODULATORS KCNK17, KCNJ2, KCNJ1 P2RY14 1272/4885FFAR2 1609/4885GLS 313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.