SCHEMBL1320875

SCHEMBL1320875

CCN(C=O)C(O)[C@H]1O[C@@H](n2cnc3c(NCc4ccccc4)ncnc32)[C@H](O)[C@@H]1O

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 8/20 0.64
TSHR P16473 2/20 0.62
TP53 P04637 1/20 0.62
SLC29A1 Q99808 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
DNPH1 O43598 1/20 0.57
PDE4A P27815 1/20 0.55
PDE4B Q07343 1/20 0.55
PDE4C Q08493 1/20 0.55
PDE4D Q08499 1/20 0.55
DOT1L Q8TEK3 1/20 0.55
DNMT1 P26358 1/20 0.55
DNMT3B Q9UBC3 1/20 0.55
NT5E P21589 1/20 0.54
CYP3A4 P08684 1/20 0.54
NFKB1 P19838 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6636036 0.85 ADORA2A (0.52) ADORA3
SCHEMBL918591 0.82 ADORA3 (0.69) ADORA3TSHRTP53SLC29A1TDP1
SCHEMBL5859134 0.82 ADORA3 (0.68) ADORA3TSHRCYP3A4NFKB1BLM
SCHEMBL5685741 0.82 ADORA2A (0.61) ADORA3TSHRTP53SLC29A1TDP1
SCHEMBL7744261 0.81 AHCY (0.46)
SCHEMBL7161647 0.81 ADORA2A (0.63) ADORA3TSHRTP53SLC29A1TDP1
SCHEMBL29877256 0.81 AHCY (0.61) ADORA3TSHRDOT1LBLM
SCHEMBL177772 0.81 AHCY (0.61) ADORA3TSHRDOT1LBLM
SCHEMBL28901883 0.81 AHCY (0.61) ADORA3TSHRDOT1LBLM
SCHEMBL27437734 0.80 ADORA3 (0.76) ADORA3TSHRTP53SLC29A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8058243-B2 Method for treating a brain cancer with ifenprodil HSC RESEARCH AND DEVELOPMENT LIMITED PARTNERSHIP (CA) 2011-11-15 US disclosed
US-20090076019-A1 METHODS FOR TREATING NEUROLOGICAL DISORDERS OR DAMAGE MOUNT SINAI HOSPITAL (CA) 2009-03-19 US disclosed