SCHEMBL13225445

SCHEMBL13225445

CNC(=O)Oc1ccc(C(=O)NOCOC)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 3/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
LMNA P02545 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MMP13 P45452 1/20 0.40
KMT2A Q03164 1/20 0.39
MAPT P10636 1/20 0.39
POLB P06746 1/20 0.39
MGLL Q99685 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12893239 0.79 HPGD (0.68) PLK1CA1CA2HPGDTSHR
SCHEMBL12418676 0.79 PLK1 (0.49) PLK1NPC1RAB9ACA1CA2
SCHEMBL12418675 0.78 ALDH1A1 (0.44) PLK1NPC1RAB9AHPGDHTT
SCHEMBL7806735 0.76 NPC1 (0.61) NPC1RAB9ACA1HPGDTSHR
SCHEMBL12680144 0.75 ALDH1A1 (0.71) NPC1RAB9AHPGDSMN1; SMN2L3MBTL1
SCHEMBL277445 0.75 PLK1 (0.51) PLK1NPC1RAB9AHPGDTSHR
SCHEMBL12893245 0.75 ALDH1A1 (0.51) PLK1NPC1RAB9AHPGDTSHR
SCHEMBL14864017 0.74 HPGD (0.60) PLK1RAB9AHPGDHTTLMNA
SCHEMBL12417397 0.73 MAPT (0.51) PLK1RAB9AMAPTALDH1A1
SCHEMBL12414159 0.73 MMP13 (0.61) PLK1NPC1RAB9ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293869-B2 Polymer conjugates of GLP-1 NEKTAR THERAPEUTICS (US) 2012-10-23 US disclosed
US-20100210505-A1 POLYMER CONJUGATES OF GLP-1 NEKTAR THERAPEUTICS AL, CORPORATION (US) 2010-08-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100210505-A1 POLYMER CONJUGATES OF GLP-1 GLP1R, GIPR, NGLY1 PLK1 2786/4885NPC1 3626/4885RAB9A 1283/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.