Eucatropine

Eucatropine

SCHEMBL132347

CC1CC(OC(=O)C(O)c2ccccc2)CC(C)(C)N1C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 1.00
LMNA P02545 5/20 0.98
NR1I2 O75469 1/20 0.65
ABCB11 O95342 1/20 0.65
CYP2C9 P11712 1/20 0.58
HSD17B10 Q99714 1/20 0.58
CHRM1 P11229 8/20 0.57
CHRM2 P08172 7/20 0.57
CHRM3 P20309 7/20 0.57
CHRM4 P08173 6/20 0.57
CHRM5 P08912 6/20 0.57
BLM P54132 2/20 0.57
TDP1 Q9NUW8 2/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
TSHR P16473 2/20 0.41
NFKB1 P19838 2/20 0.41
CYP1A2 P05177 1/20 0.41
HIF1A Q16665 1/20 0.41
HTR2C P28335 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eucatropine SCHEMBL636552 0.99 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Eucatropine SCHEMBL28210942 0.95 CYP2D6 (0.91) CYP2D6LMNANR1I2ABCB11CYP2C9
Cyclandelate SCHEMBL8060819 0.79 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Cyclandelate SCHEMBL5123 0.79 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Cyclandelate SCHEMBL547043 0.79 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Homatropine SCHEMBL23468168 0.74 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Homatropine SCHEMBL9653008 0.74 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Homatropine SCHEMBL15275620 0.74 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Homatropine SCHEMBL23970 0.74 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9
Homatropine SCHEMBL23969 0.74 LMNA (1.00) CYP2D6LMNANR1I2ABCB11CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2123 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724079-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2026-04-15 EP claimed
US-20260048096-A1 METHODS AND COMPOSITIONS FOR PRESERVING THE RETINAL OUTER NUCLEAR LAYER (ONL), PHOTORECEPTORS, AND RETINAL THICKNESS STEALTH BIOTHERAPEUTICS INC. (US) 2026-02-19 US claimed
EP-4596049-A2 PEPTIDE FOR USE IN PREVENTING OR TREATING MACULAR DEGENERATION Stealth BioTherapeutics Inc. (US) 2025-08-06 EP claimed
EP-4302829-B1 PEPTIDE FOR USE IN PREVENTING OR TREATING MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC (US) 2025-05-21 EP claimed
US-20250090621-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2025-03-20 US claimed
WO-2024254164-A2 METHODS AND COMPOSITIONS FOR THE TREATMENT OF AGE-RELATED MACULAR DEGENERATION STEALTH BIOTHERAPEUTICS INC. (US) 2024-12-12 WO claimed
US-20240350577-A1 METHODS AND COMPOSITIONS FOR PREVENTING OR TREATING DOMINANT OPTIC ATROPHY STEALTH BIOTHERAPEUTICS INC. (US) 2024-10-24 US claimed
EP-3413872-B1 NON-INVASIVE OCULAR DRUG DELIVERY INSERT TECHNOLOGY UNIV DE COIMBRA (PT) 2024-10-02 EP claimed
EP-4419123-A1 METHODS AND COMPOSITIONS COMPRISING PEPTIDOMIMITICS FOR TREATING, PREVENTING, INHIBITING, AMELIORATING OR DELAYING THE ONSET OF OPHTHALMIC CONDITIONS Stealth BioTherapeutics Inc. (US) 2024-08-28 EP claimed
WO-2024163315-A2 DERIVATIZED COLLAGEN-HYALURONIC ACID BASED IMPLANTS FOR SUSTAINED DELIVERY OF OPHTHALMIC DRUGS DEVORE DALE (US) 2024-08-08 WO claimed
EP-0126684-B1 DRUG DELIVERY SYSTEM UTILIZING THERMOSETTING GELS MERCK & CO. INC. (US) 1991-08-28 EP claimed
US-4720494-A Anticholinergic eucatropine esters and antiperspirant use thereof THE GILLETTE COMPANY (US) 1988-01-19 US claimed
US-4546096-A Anticholinergic glucuronides and antiperspirant use thereof REPLIGEN CORPORATION (US) 1985-10-08 US claimed
EP-0154446-A2 Anti-cholinergic glucuronides and their anti-perspirant use REPLIGEN CORPORATION (US) 1985-09-11 EP claimed
EP-0126684-A2 Drug delivery system utilizing thermosetting gels MERCK & CO. INC. (US) 1984-11-28 EP claimed
US-4474751-A SUSTAINED RELEASE USING AN ALKYLENEDIAMINE-MODIFIED ETHYLENE OXIDE-PROPYLENE OXIDE COPOLYMER MERCK & CO., INC. (US) 1984-10-02 US claimed
US-4186184-A Selective administration of drug with ocular therapeutic system ALZA CORPORATION (US) 1980-01-29 US claimed
US-4186185-A Compositions comprising arylene substituted poly(orthoesters) containing useful agents ALZA CORPORATION (US) 1980-01-29 US claimed
US-4066747-A Polymeric orthoesters housing beneficial drug for controlled release therefrom ALZA CORPORATION (US) 1978-01-03 US claimed
US-4014335-A Ocular drug delivery device ALZA CORPORATION (US) 1977-03-29 US claimed