Cyclandelate

Cyclandelate

SCHEMBL5123

CC1CC(OC(=O)C(O)c2ccccc2)CC(C)(C)C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 1.00
NR1I2 O75469 1/20 1.00
ABCB11 O95342 1/20 1.00
CYP2D6 P10635 3/20 0.65
CYP2C9 P11712 4/20 0.57
CYP3A4 P08684 2/20 0.57
ALDH1A1 P00352 2/20 0.57
CYP1A2 P05177 2/20 0.57
CYP2C19 P33261 1/20 0.57
HSD17B10 Q99714 2/20 0.55
CHRM2 P08172 8/20 0.54
CHRM1 P11229 7/20 0.54
CHRM3 P20309 7/20 0.54
CHRM5 P08912 6/20 0.54
CHRM4 P08173 5/20 0.54
BLM P54132 4/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
KMT2A Q03164 4/20 0.43
PABPC1 P11940 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclandelate SCHEMBL547043 1.00 LMNA (1.00) LMNANR1I2ABCB11CYP2D6CYP2C9
Cyclandelate SCHEMBL8060819 1.00 LMNA (1.00) LMNANR1I2ABCB11CYP2D6CYP2C9
Cyclandelate SCHEMBL9705893 0.86 LMNA (0.74) LMNANR1I2ABCB11CYP2D6CYP2C9
Cyclandelate SCHEMBL9705887 0.84 LMNA (0.70) LMNANR1I2ABCB11CYP2D6CYP2C9
Eucatropine SCHEMBL132347 0.79 CYP2D6 (1.00) LMNANR1I2ABCB11CYP2D6CYP2C9
SCHEMBL13894203 0.78 LMNA (0.71) LMNANR1I2ABCB11CYP2C9CYP3A4
Eucatropine SCHEMBL636552 0.78 LMNA (1.00) LMNANR1I2ABCB11CYP2D6CYP2C9
SCHEMBL6908933 0.77 ALDH1A1 (0.84) LMNANR1I2ABCB11CYP2D6CYP2C9
SCHEMBL3846512 0.77 ALDH1A1 (0.84) LMNANR1I2ABCB11CYP2D6CYP2C9
SCHEMBL3846508 0.77 ALDH1A1 (0.84) LMNANR1I2ABCB11CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4749 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
US-20260001942-A1 TREATMENT OF HEADACHE DISORDERS AND/OR PSYCHIATRIC SYMPTOMS USING ANTI-CGRP ANTIBODIES, AND COMPOSITIONS AND METHODS RELATED THERETO H LUNDBECK AS (DK) 2026-01-01 US claimed
WO-2025262247-A1 TREATMENT OF HEADACHE DISORDERS AND/OR PSYCHIATRIC SYMPTOMS USING ANTI-CGRP ANTIBODIES, AND COMPOSITIONS AND METHODS RELATED THERETO H. LUNDBECK A/S (DK) 2025-12-26 WO claimed
US-20250268841-A1 Trans-Epithelial Membrane Drug Delivery System Masiz, John J. (US) 2025-08-28 US claimed
US-20250120907-A1 Transmucosal Drug Delivery System Masiz, John J. (US) 2025-04-17 US claimed
US-12246098-B2 Trans-epithelial membrane drug delivery system BioPhysics Pharma, Inc. (US) 2025-03-11 US claimed
CN-118736809-A Flexible bus dynamic scheduling method considering hybrid request and fairness 华南理工大学 2024-10-01 CN claimed
US-12102653-B2 Ligand regulated protein-protein interaction system ST. ANNA KINDERKREBSFORSCHUNG (AT) 2024-10-01 US claimed
US-20240216292-A1 Trans-Epithelial Membrane Drug Delivery System Masiz, John J. (US) 2024-07-04 US claimed
US-20240108588-A1 Transdermal Drug Delivery System Masiz, John J. (US) 2024-04-04 US claimed
US-4769236-A Medicaments with a high degree of solubility and method for their production ELAN CORPORATION, PLC (IE) 1988-09-06 US claimed
US-4751241-A POLYGLYCEROL ESTER OF UNSATURATED FATTY ACID FREUND INDUSTRIAL COMPANY, LTD. (JP) 1988-06-14 US claimed
CN-87103560-A Pharmaceutical composition 1988-05-18 CN claimed
WO-1987005505-A1 PHARMACEUTICAL COMPOSITIONS EURASIAM LABORATORIES, INC. (US) 1987-09-24 WO claimed
US-RE32393-E STABLE, OIL IN WATER EMULSION KABIVITRUM AB (SE) 1987-04-07 US claimed
EP-0181966-A1 Compression-coated dispersible tablets GIST-BROCADES N.V. (NL) 1986-05-28 EP claimed
EP-0181650-A1 Compression-coated dispersible tablets GIST-BROCADES N.V. (NL) 1986-05-21 EP claimed
US-4555398-A THERMOSETTING OR THERMOPLASTIC RESIN MOLD CHISSO CORPORATION (JP) 1985-11-26 US claimed
US-4369172-A Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose FOREST LABORATORIES INC. (US) 1983-01-18 US claimed
US-4168308-A Composition for enhancing the administration of pharmacologically active agents APOTEKSVARUCENTRALEN VITRUM AB (SE) 1979-09-18 US claimed