SCHEMBL13246730

SCHEMBL13246730

CC(C)(C)C(=O)/C=C/c1ccc(-c2ccccc2)cc1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.69
NPC1 O15118 2/20 0.69
KMT2A Q03164 2/20 0.69
LMNA P02545 2/20 0.69
MEN1 O00255 1/20 0.69
RAB9A P51151 1/20 0.69
L3MBTL1 Q9Y468 1/20 0.69
HDAC2 Q92769 3/20 0.59
TSHR P16473 1/20 0.57
EGFR P00533 1/20 0.49
GLA P06280 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TRPM2 O94759 1/20 0.48
LTB4R Q15722 1/20 0.48
HDAC1 Q13547 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
MAPT P10636 2/20 0.47
CYP1A2 P05177 2/20 0.47
HDAC3 O15379 1/20 0.47
TNKS O95271 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047363 0.89 NPC1 (0.72) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL6047364 0.89 NPC1 (0.72) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL22951391 0.89 NPC1 (0.72) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL3136872 0.87 KMT2A (0.68) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL4821062 0.87 KMT2A (0.68) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL9422510 0.80 KMT2A (0.61) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL1284286 0.79 RAB9A (0.60) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL21235162 0.79 TYR (0.61) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL1284284 0.79 RAB9A (0.60) ALDH1A1NPC1KMT2ALMNAMEN1
SCHEMBL4054009 0.79 GLA (0.77) ALDH1A1LMNAHDAC2GLATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150337013-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS MERCK SHARP & DOHME CORP. (US) 2015-11-26 US disclosed
US-20140073558-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CUBIST PHARMACEUTICALS, INC. (US) 2014-03-13 US disclosed
US-8507647-B2 Antibacterial agents for the treatment of gram positive infections CUBIST PHARMACEUTICALS, INC. (US) 2013-08-13 US disclosed
US-20100184649-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CUBIST PHARMACEUTICALS, INC. 2010-07-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150337013-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CLPP, CLPTM1, RPN1 ALDH1A1 4703/4885NPC1 2676/4885KMT2A 4671/4885
US-20100184649-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CLPP, CLPTM1, RPN1 ALDH1A1 4703/4885NPC1 2676/4885KMT2A 4671/4885
US-20140073558-A1 NOVEL ANTIBACTERIAL AGENTS FOR THE TREATMENT OF GRAM POSITIVE INFECTIONS CLPP, CLPTM1, RPN1 ALDH1A1 4703/4885NPC1 2676/4885KMT2A 4671/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.