SCHEMBL13285202

SCHEMBL13285202

Cc1nnc2n1-c1ccccc1C(c1ccc(F)cc1)=NC2

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.77
GABRA1 P14867 9/20 0.60
GABRA5 P31644 9/20 0.60
GABRA2 P47869 9/20 0.60
GABRB2 P47870 8/20 0.60
GABRA3 P34903 6/20 0.60
OPRK1 P41145 2/20 0.60
HPGD P15428 2/20 0.60
LMNA P02545 2/20 0.60
CNR1 P21554 1/20 0.60
PTAFR P25105 5/20 0.57
GABRG2 P18507 1/20 0.53
HTR2A P28223 1/20 0.53
GABRB3 P28472 1/20 0.53
ADRA1A P35348 1/20 0.53
PDE4D Q08499 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
TSHR P16473 1/20 0.51
ALDH1A1 P00352 1/20 0.47
BRD2 P25440 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7324237 0.89 BRD4 (0.81) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL13285201 0.87 GABRA5 (0.63) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL20463079 0.85 BRD4 (0.74) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL2615310 0.85 GABRA1 (0.74) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL11730100 0.84 PTAFR (0.76) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL23881599 0.82 PTAFR (0.63) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL14215363 0.81 BRD4 (0.68) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL2615308 0.81 BRD4 (0.52) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL11620188 0.79 PTAFR (0.79) BRD4GABRA1GABRA5GABRA2GABRB2
SCHEMBL8274469 0.79 GABRA1 (0.80) BRD4GABRA1GABRA5GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010081036-A2 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-07-15 WO disclosed