SCHEMBL13324028

SCHEMBL13324028

CS(C)(Br)CC(=O)CCC(NC(=O)C(CO)NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 1/20 0.47
CASP1 P29466 1/20 0.47
CASP3 P42574 1/20 0.47
CASP7 P55210 1/20 0.47
CASP9 P55211 1/20 0.47
MME P08473 3/20 0.46
ECE1 P42892 3/20 0.46
ACE P12821 1/20 0.46
CTSL P07711 2/20 0.46
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
FOLH1 Q04609 1/20 0.45
CTSK P43235 2/20 0.44
CAPN1 P07384 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13324027 0.92 CASP1 (0.55) CASP1CASP3CASP7CASP9MME
SCHEMBL13324023 0.92 ACE (0.54) ACECTSLCTSKCAPN1
SCHEMBL13324016 0.90 MME (0.54) CASP1CASP3CASP7CASP9MME
SCHEMBL13324026 0.89 CTSK (0.49) PSMB5CASP1CASP3CASP7CASP9
SCHEMBL13324022 0.89 CASP3 (0.55) CASP1CASP3CASP7CASP9MME
SCHEMBL13324032 0.88 ACE (0.57) MMEECE1ACECTSLSIRT2
SCHEMBL13324008 0.86 MME (0.50) MMEECE1ACECTSLSIRT2
SCHEMBL13324029 0.86 SIRT2 (0.49) CASP1CASP3CASP7CASP9MME
SCHEMBL13324031 0.85 ITGB3 (0.51) CASP1CASP3CASP7CASP9ACE
SCHEMBL13324018 0.85 CASP3 (0.56) PSMB5CASP1CASP3CASP7CASP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7723307-B2 Amino acid derivatives and pharmaceutical uses thereof ASTON UNIVERSITY (GB) 2010-05-25 US disclosed
US-20080200511-A1 Novel Compounds and Methods of Using the Same ASTON UNIVERSITY (GB) 2008-08-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080200511-A1 Novel Compounds and Methods of Using the Same F3, IL4I1, TPMT PSMB5 1249/4885CASP1 709/4885CASP3 1245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.