SCHEMBL13384451

SCHEMBL13384451

CCn1c(=O)[nH]cc(C(C)C)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.39
PDE4A P27815 4/20 0.39
PDE4B Q07343 4/20 0.39
PDE4C Q08493 4/20 0.39
PDE4D Q08499 4/20 0.39
CYP1A2 P05177 3/20 0.38
BTK Q06187 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSP90AA1 P07900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13384452 0.78 SLC9A1 (0.47) ADRA1AADRA1BLMNAHSP90AA1SLC9A1
SCHEMBL7521745 0.77 ALDH1A1 (0.48) MEN1KMT2ACYP3A4SMN1; SMN2HSP90AA1
SCHEMBL14639338 0.75 ADORA2A (0.42) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL15614498 0.75 ADORA2B (0.34) ADORA2AADRA1AADRA1BLMNACYP3A4
SCHEMBL8876920 0.75 SLC9A1 (0.53) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL12657637 0.73 ADORA2A (0.41) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL16503636 0.73 ALDH1A1 (0.35) ADORA2BDAOALDH1A1
SCHEMBL27989701 0.73 CYP1A2 (0.51) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL3581221 0.70
SCHEMBL19723176 0.69 ALDH1A1 (0.35) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7696210-B2 Gonadotropin releasing hormone receptor antagonists WYETH (US) 2010-04-13 US disclosed