SCHEMBL7521745

SCHEMBL7521745

CC(C)c1c[nH]c(=O)n(Cc2ccccc2)c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.48
HPGD P15428 4/20 0.48
KDM4E B2RXH2 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TLR7 Q9NYK1 2/20 0.45
USP1 O94782 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
P2RX4 Q99571 1/20 0.41
HSP90AA1 P07900 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
CYP3A4 P08684 1/20 0.41
LGMN Q99538 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2B P29275 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PNP P00491 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4098207 0.80 MEN1 (0.53) ALDH1A1HPGDKDM4ESMN1; SMN2TLR7
SCHEMBL13384451 0.77 ADORA2A (0.39) ALDH1A1SMN1; SMN2HSP90AA1CYP3A4ADORA2B
SCHEMBL4164688 0.76 ALDH1A1 (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
SCHEMBL1584775 0.76 ALDH1A1 (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
SCHEMBL27422649 0.76 ALDH1A1 (0.49) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
SCHEMBL11315740 0.75 HPGD (0.50) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
SCHEMBL15978138 0.75 FPR1 (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
Hydrogen Sulfide SCHEMBL27583639 0.75 HPGD (0.50) ALDH1A1HPGDKDM4ESMN1; SMN2P2RX4
SCHEMBL7844750 0.73 HPGD (0.51) ALDH1A1HPGDKDM4ESMN1; SMN2TLR7
SCHEMBL3993882 0.73 KDM4E (0.48) ALDH1A1HPGDKDM4ESMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1169310-A1 PROCESS FOR PREPARING MKC-442 Triangle Pharmaceuticals Inc. (US) 2002-01-09 EP disclosed
WO-2000061566-A1 PROCESS FOR PREPARING MKC-442 TRIANGLE PHARMACEUTICALS, INC. (US) 2000-10-19 WO disclosed