SCHEMBL13475308

SCHEMBL13475308

CCCc1cc(S(=O)(=O)C(F)(F)F)ccc1NC(=O)c1c(C)c(-c2ccc(C#N)cc2)cc(C(C)(C)C)c1O

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.34
LMNA P02545 2/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
METAP2 P50579 1/20 0.33
NR1H2 P55055 1/20 0.32
NR1H3 Q13133 1/20 0.32
EPAS1 Q99814 1/20 0.32
PTGFR P43088 1/20 0.32
TSHR P16473 1/20 0.31
BRAF P15056 1/20 0.31
SLC22A12 Q96S37 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13475304 0.94 HSD11B1 (0.34) HSD11B1LMNAALDH1A1SMN1; SMN2NR1H2
SCHEMBL13475303 0.89 NR1H2 (0.34) HSD11B1LMNAALDH1A1SMN1; SMN2NR1H2
SCHEMBL13475305 0.88 EPAS1 (0.35) HSD11B1NR1H2NR1H3EPAS1PTGFR
SCHEMBL13475213 0.87 NR1H2 (0.42) HSD11B1LMNAALDH1A1SMN1; SMN2NR1H2
SCHEMBL2788779 0.83 MEN1 (0.41) LMNAALDH1A1SMN1; SMN2METAP2PTGFR
SCHEMBL13475208 0.78 CA1 (0.42) MEN1KMT2A
SCHEMBL13475218 0.77 PDK1 (0.45) MEN1KMT2A
SCHEMBL2789511 0.76 MEN1 (0.43) LMNAALDH1A1SMN1; SMN2PTGFRTSHR
SCHEMBL13475315 0.76 KMT2A (0.41) LMNANR1H2NR1H3PTGFRMEN1
SCHEMBL13436115 0.76 GCGR (0.38) PTGFRSLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100041657-A1 HALOALKYLSULFONE SUBSTITUTED COMPOUNDS USEFUL FOR TREATING OBESITY AND DIABETES NOVO NORDICK A/S (DK) 2010-02-18 US disclosed
US-20100041657-A1 HALOALKYLSULFONE SUBSTITUTED COMPOUNDS USEFUL FOR TREATING OBESITY AND DIABETES NOVO NORDICK A/S (DK) 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100041657-A1 HALOALKYLSULFONE SUBSTITUTED COMPOUNDS USEFUL FOR TREATING OBESITY AND DIABETES RPS12, GPR119, ATP12A HSD11B1 66/4885LMNA 4278/4885ALDH1A1 899/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.