SCHEMBL13484115

SCHEMBL13484115

COc1ccc2cc(C=C(C)C)ccc2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.50
CYP2A6 P11509 1/20 0.50
NQO2 P16083 4/20 0.47
PTGS2 P35354 5/20 0.47
PTGS1 P23219 3/20 0.47
KDM4E B2RXH2 2/20 0.47
CYP1A1 P04798 2/20 0.47
CYP1B1 Q16678 2/20 0.47
LMNA P02545 1/20 0.47
ALOX12 P18054 1/20 0.47
MAOB P27338 1/20 0.47
RELA Q04206 2/20 0.46
ESR1 P03372 2/20 0.46
ABL1 P00519 1/20 0.46
TTR P02766 1/20 0.46
ABCB1 P08183 1/20 0.46
ALOX5 P09917 1/20 0.46
BCR P11274 1/20 0.46
CYP19A1 P11511 1/20 0.46
TUBB4A P04350 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7345665 0.83 RELA (0.49) CYP1A2CYP2A6NQO2PTGS2PTGS1
SCHEMBL7334386 0.83 PLAU (0.44) CYP1A2CYP2A6NQO2MAOBRELA
SCHEMBL7334384 0.83 PLAU (0.44) CYP1A2CYP2A6NQO2MAOBRELA
SCHEMBL21470094 0.82 MAOB (0.49) CYP1A2CYP2A6NQO2KDM4ELMNA
SCHEMBL13484378 0.82 NQO2 (0.45) CYP1A2CYP2A6NQO2PTGS2PTGS1
SCHEMBL14325968 0.82 MAOB (0.46) CYP1A2CYP2A6NQO2PTGS2PTGS1
SCHEMBL12169007 0.81 ALDH1A1 (0.63) CYP1A2CYP2A6NQO2PTGS2PTGS1
SCHEMBL7158461 0.79 MAPT (0.72) CYP1A2CYP2A6NQO2KDM4ELMNA
SCHEMBL14303313 0.79 EGFR (0.56) CYP1A2PTGS2PTGS1KDM4ELMNA
SCHEMBL28673144 0.79 EGFR (0.56) CYP1A2PTGS2PTGS1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8337941-B2 Fluorescent substrates for monoamine transporters as optical false neurotransmitters THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2012-12-25 US disclosed
US-20100035279-A1 Fluorescent Substrates for Monoamine Transporters as Optical False Neurotransmitters NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2010-02-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100035279-A1 Fluorescent Substrates for Monoamine Transporters as Optical False Neurotransmitters SLC18A2, SLC6A2, SLC18A3 CYP1A2 1053/4885CYP2A6 1899/4885NQO2 248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.