SCHEMBL135288

SCHEMBL135288

O=C(O)C1=NOC(c2ccccc2)(c2ccccc2)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.35
HDAC9 Q9UKV0 1/20 0.34
POLB P06746 1/20 0.33
HSD11B1 P28845 2/20 0.33
HCAR3 P49019 1/20 0.33
HCAR2 Q8TDS4 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP1A2 P05177 1/20 0.33
HDAC4 P56524 2/20 0.33
CHRM2 P08172 3/20 0.32
CHRM4 P08173 3/20 0.32
CHRM5 P08912 3/20 0.32
CHRM1 P11229 3/20 0.32
CHRM3 P20309 3/20 0.32
LDHA P00338 1/20 0.32
LDHB P07195 1/20 0.32
CA1 P00915 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1832298 0.91 PTGDR2 (0.38) POLBHSD11B1HCAR3HCAR2MEN1
Isopropylamine SCHEMBL28970090 0.91 ALDH1A1 (0.34) HCAR3HCAR2MEN1KMT2ACYP1A2
SCHEMBL28574647 0.86 POLB (0.35) AKR1C1HDAC9POLBHSD11B1MEN1
SCHEMBL29498824 0.86 LDHA (0.36) AKR1C1HDAC9HSD11B1MEN1NPC1
SCHEMBL7167294 0.82 MAPT (0.45) MEN1RAB9AKMT2ACYP1A2TSHR
SCHEMBL12971595 0.82 HDAC4 (0.31) HDAC4
SCHEMBL27915985 0.82 CA1 (0.38) HDAC9POLBHCAR2NPC1RAB9A
SCHEMBL28970097 0.80 MAPT (0.43) KMT2ACHRM2CHRM1TSHRALDH1A1
SCHEMBL31501098 0.79 MEN1 (0.37) AKR1C1HDAC9POLBHSD11B1HCAR3
SCHEMBL31501097 0.79 MEN1 (0.37) AKR1C1HDAC9POLBHSD11B1HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8308 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3947350-B1 SUBSTITUTED 2-HETEROARYL AMINOBENZENES, THEIR SALTS AND USE OF SAID COMPOUNDS AS HERBICIDAL AGENTS BAYER AG (DE) 2026-05-27 EP claimed
EP-4742896-A1 HERBICIDE COMPOSITIONS COMPRISING MALONAMIDES AND SAFENERS FOR SELECTIVE WEED CONTROL IN CROPS BASF SE (DE) 2026-05-20 EP claimed
WO-2026088192-A1 METHOD FOR CONTROLLING WEED IN CEREAL CROPS ADAMA AGAN LTD. (IL) 2026-04-30 WO claimed
US-12610950-B2 Method for weed control in lawn or turf DISCOVERY PURCHASER CORPORATION (US) 2026-04-28 US claimed
US-20260096553-A1 MICROENCAPSULATED HERBICIDES MONSANTO TECHNOLOGY LLC (US) 2026-04-09 US claimed
US-20260076368-A1 HERBICIDAL COMPOSITION COMPRISING BIFENOX AND VLCFA INHIBITOR ADAMA AGAN LTD. (IL) 2026-03-19 US claimed
US-20260068883-A1 PROTOPORPHYRINOGEN OXIDASE INHIBITORS ENKO CHEM, INC. (US) 2026-03-12 US claimed
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
EP-4658060-A1 GENERATING DOUBLED HAPLOID PLANTS Syngenta Crop Protection AG (CH) 2025-12-10 EP claimed
US-20250359550-A1 METHOD FOR WEED CONTROL IN LAWN OR TURF DISCOVERY PURCHASER CORPORATION (US) 2025-11-27 US claimed
EP-1306007-A1 Compositions and method to safen crops from injury caused by uracil-substituted benzisothiazoles BASF AKTIENGESELLSCHAFT (DE) 2003-05-02 EP claimed
WO-2003028460-A2 HERBICIDAL COMPOSITION SYNGENTA PARTICIPATIONS AG (CH) 2003-04-10 WO claimed
WO-2003024221-A1 HERBICIDAL MIXTURES BASED ON 3-PHENYLURACILS BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO claimed
WO-2002100171-A1 HERBICIDAL COMPOSITION SYNGENTA PARTICIPATIONS AG (CH) 2002-12-19 WO claimed
CN-1378424-A Selective herbicides on basis of n-aryl-trizoline (thio) ones BAYER AG (DE) 2002-11-06 CN claimed
WO-2002060256-A1 METHOD OF SAFENING CROPS USING ISOXAZOLINE CARBOXYLATES BAYER CROPSCIENCE GMBH (DE) 2002-08-08 WO claimed
WO-2002060255-A2 HERBICIDE-SAFENER COMBINATION BASED ON ISOXOZOLINE CARBOXYLATE SAFENERS BAYER CROPSCIENCE GMBH (DE) 2002-08-08 WO claimed
EP-1213966-A1 NEW HERBICIDAL COMPOSITIONS Bayer CropScience Limited (GB) 2002-06-19 EP claimed
WO-2001043546-A2 COMBINATIONS OF HERBICIDAL ALKYLAZINES AND SAFENERS AVENTIS CROPSCIENCE GMBH (DE) 2001-06-21 WO claimed
WO-2001017350-A1 NEW HERBICIDAL COMPOSITIONS AVENTIS CROPSCIENCE UK LIMITED (GB) 2001-03-15 WO claimed