SCHEMBL13612049

SCHEMBL13612049

COc1ccccc1CNC(=O)C1CN2C(=N1)N=C(C)C(CN)=C2c1ccc(Cl)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 1/20 0.40
ANO2 Q9NQ90 1/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 1/20 0.39
SMO Q99835 1/20 0.39
HPGD P15428 2/20 0.39
HTT P42858 1/20 0.39
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
DRD2 P14416 1/20 0.37
DRD1 P21728 1/20 0.37
EPHX2 P34913 1/20 0.37
DPP4 P27487 2/20 0.37
DPP8 Q6V1X1 1/20 0.37
DPP9 Q86TI2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13612023 0.88 ALDH1A1 (0.38) CYP3A4ALDH1A1HTTLMNATSHR
SCHEMBL13611767 0.83 TDP1 (0.38) CYP3A4CYP2C19ALDH1A1EPHX2DPP4
SCHEMBL13611864 0.79 DPP4 (0.40) CYP3A4CYP2C19ALDH1A1MEN1KMT2A
SCHEMBL13611902 0.77 DPP4 (0.46) SMOEPHX2DPP4DPP8DPP9
SCHEMBL13612016 0.76 DPP4 (0.44) MEN1KMT2ADPP4DPP8DPP9
SCHEMBL13612029 0.73 DPP4 (0.48) SMOMEN1KMT2ADRD2DPP4
SCHEMBL13611869 0.73 DPP4 (0.36) MAPTDPP4DPP8DPP9
SCHEMBL13612007 0.72 DPP4 (0.35) CYP3A4CYP2C9CYP2C19DPP4DPP8
SCHEMBL13308028 0.65 CNR1 (0.77) ANO1ANO2CYP3A4CYP2C9CYP2C19
SCHEMBL8257313 0.64 DPP4 (0.70) DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7635699-B2 Azolopyrimidine-based inhibitors of dipeptidyl peptidase IV and methods BRISTOL-MYERS SQUIBB COMPANY (US) 2009-12-22 US disclosed