SCHEMBL13612029

SCHEMBL13612029

COC[C@H]1CCCN1C(=O)C1CN2C(=N1)N=C(C)C(CN)=C2c1ccc(Cl)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.48
DPP8 Q6V1X1 4/20 0.48
DPP9 Q86TI2 2/20 0.48
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNB3 Q05901 1/20 0.35
CHRM3 P20309 1/20 0.35
SMO Q99835 1/20 0.34
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
KCNH2 Q12809 1/20 0.33
BACE1 P56817 1/20 0.32
KMT2A Q03164 2/20 0.32
ENPP2 Q13822 2/20 0.32
MET P08581 1/20 0.32
ADORA2A P29274 4/20 0.32
CAMK1D Q8IU85 1/20 0.32
FPR1 P21462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13611879 1.00 DPP4 (0.48) DPP4DPP8DPP9CHRNB1CHRNB2
SCHEMBL13612016 0.84 DPP4 (0.44) DPP4DPP8DPP9KMT2AMEN1
SCHEMBL13612014 0.79 MAPT (0.40) DPP4DPP8DPP9KMT2AMEN1
SCHEMBL13611869 0.79 DPP4 (0.36) DPP4DPP8DPP9
SCHEMBL13612018 0.76 DPP4 (0.50) DPP4DPP8DPP9SMO
SCHEMBL13611902 0.75 DPP4 (0.46) DPP4DPP8DPP9SMO
SCHEMBL13612023 0.74 ALDH1A1 (0.38) DPP4DPP8DPP9KMT2AMEN1
SCHEMBL13612028 0.74 MEN1 (0.36) DPP4DPP8CHRM3KMT2AMEN1
SCHEMBL13612049 0.73 ANO1 (0.40) DPP4DPP8DPP9SMODRD2
SCHEMBL13612035 0.73 MAPT (0.41) DPP4KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7635699-B2 Azolopyrimidine-based inhibitors of dipeptidyl peptidase IV and methods BRISTOL-MYERS SQUIBB COMPANY (US) 2009-12-22 US disclosed