SCHEMBL13613558

SCHEMBL13613558

COC(=O)c1ccc(C(C#N)C(N)=O)c([N+](=O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 1/20 0.40
ALDH1A1 P00352 5/20 0.38
MAPT P10636 4/20 0.38
HPGD P15428 4/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
GLA P06280 1/20 0.38
GAA P10253 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
ATM Q13315 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA7 P43166 1/20 0.37
XDH P47989 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
PRSS1 P07477 1/20 0.36
ACR P10323 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL351791 0.89 VCAM1 (0.50) VCAM1ALDH1A1MAPTHPGDKMT2A
SCHEMBL13152525 0.89 VCAM1 (0.39) VCAM1ALDH1A1MAPTHPGDKDM4E
SCHEMBL15139324 0.84 ALDH1A1 (0.41) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL3214507 0.82 KDM4E (0.51) ALDH1A1MAPTHPGDKDM4EHSD17B10
SCHEMBL14236511 0.78
SCHEMBL3118623 0.74 KMT2A (0.49) VCAM1ALDH1A1MAPTHPGDKDM4E
SCHEMBL13619445 0.73 VCAM1 (0.42) VCAM1ALDH1A1MAPTHPGDKDM4E
SCHEMBL17204265 0.71 MAPT (0.47) VCAM1ALDH1A1MAPTHPGDKDM4E
SCHEMBL16254547 0.70 CA12 (0.62) VCAM1ALDH1A1MAPTHPGDKDM4E
SCHEMBL28072772 0.69 VCAM1 (0.53) VCAM1ALDH1A1MAPTHPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119703-A1 NOVEL INDOLE DERIVATIVE HAVING INHIBITORY ACTIVITY ON I B KINASE Santen Pharmaceutical Co., Ltd (JP) 2009-11-18 EP disclosed