SCHEMBL13613859

SCHEMBL13613859

COC(=O)Cc1ccc(-c2ccc3c(c2)C(C)(C)CC=C3OS(=O)(=O)C(F)(F)F)cc1F

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.34
CYP26B1 Q9NR63 1/20 0.34
ACLY P53396 1/20 0.33
RARA P10276 5/20 0.33
PDK2 Q15119 2/20 0.32
RARG P13631 5/20 0.32
RARB P10826 4/20 0.32
BDKRB1 P46663 5/20 0.31
CNR1 P21554 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4519345 0.89 RARA (0.37) CYP26A1CYP26B1RARARARGRARB
SCHEMBL17276192 0.74 PDK2 (0.33) RARAPDK2RARGRARB
SCHEMBL13613860 0.74 CYP26A1 (0.37) CYP26A1CYP26B1RARARARGRARB
SCHEMBL8433747 0.72 RARA (0.50) RARAPDK2RARGRARB
SCHEMBL8772764 0.71 RARB (0.33) RARAPDK2RARGRARB
SCHEMBL6292935 0.70 PDK2 (0.45) CYP26A1RARAPDK2RARGRARB
SCHEMBL8331635 0.69 PDK2 (0.46) RARAPDK2RARGRARB
SCHEMBL8664382 0.69 RARB (0.44) RARAPDK2RARGRARB
SCHEMBL13613862 0.69 PDK2 (0.37) CYP26A1CYP26B1RARAPDK2RARG
SCHEMBL6293844 0.68 ALDH1A1 (0.35) CYP26A1CYP26B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7638648-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN INC. (US) 2009-12-29 US disclosed
US-20080004455-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2008-01-03 US disclosed
US-7226951-B2 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same ALLERGAN, INC. (US) 2007-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004455-A1 Compounds having selective cytochrome P450RAI-1 or selective cytochrome P450RAI-2 inhibitory activity and methods of obtaining the same CYP1A2, CYP2A7, CYP3A7 CYP26A1 15/4885CYP26B1 10/4885ACLY 874/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.