SCHEMBL13617840

SCHEMBL13617840

N#Cc1cccc(-c2ccc(NC3CCN(Cc4cccnc4)CC3)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.52
MCHR1 Q99705 3/20 0.49
JAK3 P52333 2/20 0.47
PRKAA2 P54646 2/20 0.47
JAK2 O60674 2/20 0.47
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 3/20 0.46
CYP2C9 P11712 2/20 0.46
DRD4 P21917 1/20 0.46
DRD3 P35462 1/20 0.46
JAK1 P23458 2/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP1A2 P05177 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
CCR2 P41597 1/20 0.45
ROCK1 Q13464 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2425776 0.83 ROCK2 (0.56) ROCK2JAK3JAK2DRD4DRD3
SCHEMBL5631821 0.75 ACHE (0.60) ROCK2CYP3A4DRD4DRD3CCR2
SCHEMBL3311559 0.74 DRD4 (0.56) ROCK2DRD4CCR2ROCK1LMNA
SCHEMBL4237535 0.74 THRB (0.65) ROCK2PRKAA2CCR2ROCK1KDM4E
SCHEMBL14014430 0.74 MCHR1 (0.52) MCHR1
SCHEMBL1717462 0.73 ROCK2 (0.80) ROCK2CCR2ROCK1
SCHEMBL11465989 0.71 SIGMAR1 (0.62) ROCK2DRD4DRD3ALDH1A1MAPK1
SCHEMBL23251886 0.70 CHRNB2 (0.62) ROCK2DRD4ALDH1A1ROCK1LMNA
SCHEMBL4623213 0.70 CHRNB2 (0.62) ROCK2DRD4ALDH1A1ROCK1LMNA
Hydrochloric Acid SCHEMBL20553070 0.69 CHRNB2 (0.60) ROCK2DRD4ALDH1A1ROCK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339684-B1 MCH ANTAGONISTS AND THEIR USE IN THE TREATMENT OF OBESITY SCHERING CORP (US) 2009-11-04 EP disclosed