SCHEMBL13626501

SCHEMBL13626501

CN(C)C(=N)c1cccc(CNC(=O)C2Cc3ccccc3CN2C(=O)Nc2ccc(Cl)cc2)c1

nearest known ligand 0.59

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CFTR P13569 15/20 0.59
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626503 0.84 CFTR (0.56) CFTRLMNAPKM
SCHEMBL13626499 0.79 CFTR (0.48) CFTR
SCHEMBL13626527 0.75 CFTR (0.46) CFTRLMNAPKM
SCHEMBL13626534 0.74 CFTR (0.49) CFTR
SCHEMBL4558064 0.72 TAS1R3 (0.60) CFTRLMNAPKM
SCHEMBL13626543 0.71 CFTR (0.41) CFTRLMNAPKM
SCHEMBL13626492 0.71 CFTR (0.55) CFTRLMNAPKM
SCHEMBL13626517 0.70 CFTR (0.50) CFTRLMNAPKM
SCHEMBL7738204 0.70 HDAC8 (0.60)
SCHEMBL3922221 0.69 CFTR (0.76) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed