SCHEMBL13626544

SCHEMBL13626544

O=C(Nc1ccc(-c2cccc[n+]2[O-])cc1)C1c2ccccc2CN1C(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
RECQL P46063 1/20 0.41
PPARD Q03181 1/20 0.40
XIAP P98170 2/20 0.39
HSP90AA1 P07900 2/20 0.37
HSP90AB1 P08238 2/20 0.37
NAMPT P43490 1/20 0.36
CFTR P13569 2/20 0.36
F11 P03951 1/20 0.36
LHCGR P22888 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626486 0.85 CFTR (0.50) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL13626542 0.78 F10 (0.43) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL13626548 0.77 LMNA (0.46) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL4606642 0.76 F10 (0.54) TAS1R3TAS1R1TAS1R2
SCHEMBL4605212 0.76 F10 (0.54) TAS1R3TAS1R1TAS1R2
SCHEMBL13626545 0.75 F10 (0.49) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL4604029 0.72 F10 (0.42) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL4606187 0.72 F10 (0.42) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL14507138 0.72 F10 (0.54) TAS1R3TAS1R1TAS1R2MEN1KMT2A
SCHEMBL13626546 0.72 F10 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed