SCHEMBL13626486

SCHEMBL13626486

O=C(Nc1ccc(-c2cccc[n+]2[O-])cc1)C1Cc2ccccc2CN1C(=O)Nc1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CFTR P13569 9/20 0.50
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
TAS1R2 Q8TE23 1/20 0.46
LMNA P02545 1/20 0.46
PKM P14618 1/20 0.46
MEN1 O00255 1/20 0.44
GAA P10253 1/20 0.44
KMT2A Q03164 1/20 0.44
POLB P06746 2/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAPT P10636 2/20 0.43
MMP8 P22894 2/20 0.43
MMP3 P08254 1/20 0.43
CTDSP1 Q9GZU7 1/20 0.42
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13626548 0.85 LMNA (0.46) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL13626544 0.85 TAS1R3 (0.43) CFTRTAS1R3TAS1R1TAS1R2MEN1
SCHEMBL13626484 0.78 CFTR (0.49) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL13626481 0.78 CFTR (0.49) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL13626490 0.78 CFTR (0.49) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL4558064 0.77 TAS1R3 (0.60) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL13626502 0.76 LMNA (0.58) CFTRTAS1R3TAS1R1TAS1R2LMNA
SCHEMBL13626552 0.76 F10 (0.61) CFTR
SCHEMBL13626553 0.76 F10 (0.61) CFTR
SCHEMBL13626503 0.75 CFTR (0.56) CFTRTAS1R3TAS1R1TAS1R2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612089-B2 Tetrahydroisoquinolines as factor Xa inhibitors PORTOLA PHARMACEUTICALS, INC. (US) 2009-11-03 US disclosed