SCHEMBL13630907

SCHEMBL13630907

COC(=O)NCCNC(=O)C(C)(O)c1cc(F)cc(F)c1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.36
EPHX1 P07099 1/20 0.33
SYK P43405 1/20 0.33
TSHR P16473 1/20 0.32
SLC6A3 Q01959 1/20 0.32
CYP3A4 P08684 1/20 0.32
HTT P42858 1/20 0.32
SCN9A Q15858 1/20 0.31
CHRM1 P11229 1/20 0.31
MTNR1A P48039 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13630908 0.83 RECQL (0.47) HDAC6TSHR
SCHEMBL1161078 0.68 NR5A2 (0.42) HDAC6HTT
SCHEMBL3941432 0.68 CES2 (0.39) TSHRSLC6A3HTT
SCHEMBL22938122 0.68 CES2 (0.39) HDAC6SLC6A3HTT
SCHEMBL3941437 0.68 CES2 (0.39) TSHRSLC6A3HTT
SCHEMBL31194929 0.68 ALDH1A1 (0.58) EPHX1MTNR1A
SCHEMBL4151018 0.67 CNR2 (0.40) TSHRCYP3A4HTT
SCHEMBL4151017 0.67 CNR2 (0.40) TSHRCYP3A4HTT
SCHEMBL3190326 0.66 EPHX1 (0.61) EPHX1TSHR
SCHEMBL3180074 0.65 ALOX5 (0.39) HDAC6SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2119702-A1 AMIDE DERIVATIVE Dainippon Sumitomo Pharma Co., Ltd. (JP) 2009-11-18 EP disclosed