SCHEMBL13643113

SCHEMBL13643113

C[C@H](CO[Si](C)(C)C(C)(C)C)Cc1ccc(N)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TSHR P16473 2/20 0.32
SLC6A4 P31645 2/20 0.32
TP53 P04637 1/20 0.32
IDO1 P14902 2/20 0.32
ADRB2 P07550 5/20 0.31
TDP1 Q9NUW8 2/20 0.31
GFER P55789 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
ADRB1 P08588 1/20 0.31
ADRB3 P13945 1/20 0.31
EBP Q15125 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
LOXL2 Q9Y4K0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7361270 0.84 MME (0.35) NPC1RAB9ATSHRTP53IDO1
SCHEMBL7358574 0.81 LPL (0.39)
SCHEMBL133816 0.76 MAOB (0.39) NPC1RAB9ATSHRIDO1TDP1
SCHEMBL14832848 0.76 ADRB2 (0.33) NPC1RAB9AIDO1ADRB2ALDH1A1
SCHEMBL2617264 0.76 ATM (0.47) RAB9ATSHRTP53ALDH1A1CYP3A4
SCHEMBL13643112 0.74 CA1 (0.35) ALDH1A1
SCHEMBL2366928 0.73 GFER (0.45) NPC1RAB9ATSHRTP53TDP1
SCHEMBL22591638 0.73 GFER (0.50) TSHRADRB2TDP1GFERALDH1A1
SCHEMBL8076557 0.73
SCHEMBL13643110 0.73 CPB1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8772507-B2 Imidazole-benzamide anti-cancer agents CYTOKINETICS, INC. (US) 2014-07-08 US disclosed
US-20130096315-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS QIAN XIANGPING (US) 2013-04-18 US disclosed
US-20120283287-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS QIAN XIANGPING (US) 2012-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120283287-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS KIF5B, KIF2C, PLK1 NPC1 835/4885RAB9A 1213/4885TSHR 4714/4885
US-20130096315-A1 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS AND METHODS KIF5B, KIF2C, PLK1 NPC1 619/4885RAB9A 1283/4885TSHR 4746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.