SCHEMBL13660764

SCHEMBL13660764

COC(=O)c1ccc(CNC(=O)C(c2ccc(CN3N=C(c4ccccc4)CCC3=O)cc2)C2CCCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.48
LMNA P02545 1/20 0.47
KMT2A Q03164 1/20 0.47
PGR P06401 1/20 0.44
POLB P06746 2/20 0.42
HRH3 Q9Y5N1 1/20 0.42
PDE4A P27815 2/20 0.42
PDE4B Q07343 2/20 0.42
PDE4C Q08493 2/20 0.42
PDE4D Q08499 2/20 0.42
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
BDKRB2 P30411 1/20 0.41
THRB P10828 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7606111 0.92 KMT2A (0.47) TP53LMNAKMT2APGRPOLB
SCHEMBL7602899 0.92 LMNA (0.50) TP53LMNAKMT2APGRPOLB
SCHEMBL1081746 0.86 BDKRB2 (0.40) LMNAKMT2APDE4APDE4BPDE4C
SCHEMBL7604032 0.84 PGR (0.42) TP53LMNAKMT2APGRPDE4A
SCHEMBL7601937 0.82 BDKRB2 (0.37) TP53LMNAKMT2APGRHRH3
SCHEMBL7601099 0.81 KMT2A (0.45) TP53LMNAKMT2APGRPOLB
SCHEMBL7605776 0.81 KMT2A (0.47) TP53LMNAKMT2APGRPOLB
SCHEMBL7604168 0.81 KMT2A (0.48) TP53LMNAKMT2APGRPOLB
SCHEMBL7904520 0.80 KMT2A (0.46) TP53LMNAKMT2APGRPOLB
SCHEMBL1177753 0.80 MAOB (0.40) TP53PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009127338-A1 OXO-HETEROCYCLIC SUBSTITUTED CARBOXYLIC ACID DERIVATES AND THE USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-10-22 WO disclosed