SCHEMBL13680472

SCHEMBL13680472

CC(=O)c1ccc(-c2cccc(C)n2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.52
CCR8 P51685 1/20 0.52
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CYP2A6 P11509 1/20 0.50
ADORA3 P0DMS8 3/20 0.46
HSD17B1 P14061 1/20 0.46
GRM5 P41594 1/20 0.45
MAOB P27338 1/20 0.43
RAB9A P51151 2/20 0.42
BRD4 O60885 1/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
TGFBR1 P36897 1/20 0.41
PIK3CD O00329 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2346786 0.86 RARA (0.55) CCR1CCR8SMN1; SMN2CYP2A6GRM5
SCHEMBL13680552 0.84 CYP2A6 (0.53) CCR1CCR8CYP2A6GRM5BRD4
SCHEMBL29949633 0.84 TGFBR1 (0.50) CCR1CCR8CYP2A6GRM5TGFBR1
Hydrochloric Acid SCHEMBL3088531 0.84 RARA (0.54) CCR1CCR8SMN1; SMN2CYP2A6GRM5
SCHEMBL12270020 0.84 TGFBR1 (0.50) CCR1CCR8CYP2A6GRM5TGFBR1
SCHEMBL3422361 0.82 CCR1 (0.75) CCR1CCR8MAPTCYP2A6RAB9A
SCHEMBL13680667 0.82 CCR1 (0.52) CCR1CCR8MAPTCYP2A6GRM5
SCHEMBL13680501 0.81 GRM5 (0.52) CCR1CCR8MAPTSMN1; SMN2CYP2A6
SCHEMBL13680471 0.81 TDP1 (0.50) CCR1CCR8MAPTSMN1; SMN2CYP2A6
SCHEMBL13680473 0.81 TGFBR1 (0.48) CCR1CCR8SMN1; SMN2CYP2A6GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed