SCHEMBL13680473

SCHEMBL13680473

Cc1cccc(-c2ccc(C(=O)N(C)C)cc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.48
CCR1 P32246 1/20 0.47
CCR8 P51685 1/20 0.47
ALDH1A1 P00352 5/20 0.47
CYP3A4 P08684 4/20 0.47
HPGD P15428 3/20 0.47
TP53 P04637 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
CYP2D6 P10635 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HIF1A Q16665 1/20 0.47
CYP2A6 P11509 1/20 0.46
CYP1A2 P05177 5/20 0.45
CLK4 Q9HAZ1 4/20 0.45
CYP2C9 P11712 2/20 0.45
ATR Q13535 5/20 0.45
HSD17B10 Q99714 3/20 0.44
TSHR P16473 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12269983 0.86 KEAP1 (0.50) TGFBR1CCR1CCR8CYP3A4CYP2A6
SCHEMBL13680472 0.81 CCR1 (0.52) TGFBR1CCR1CCR8ALDH1A1HPGD
SCHEMBL2346786 0.81 RARA (0.55) CCR1CCR8ALDH1A1HPGDKDM4E
SCHEMBL13680670 0.81 ALDH1A1 (0.47) TGFBR1CCR1CCR8ALDH1A1HPGD
SCHEMBL15709459 0.80 ERN1 (0.47) ALDH1A1CYP3A4HPGDTP53KDM4E
SCHEMBL15349861 0.80 ALDH1A1 (0.44) ALDH1A1CYP3A4HPGDTP53KDM4E
SCHEMBL12270020 0.80 TGFBR1 (0.50) TGFBR1CCR1CCR8CYP2A6GRM5
Hydrochloric Acid SCHEMBL3088531 0.80 RARA (0.54) CCR1CCR8ALDH1A1HPGDKDM4E
SCHEMBL29949633 0.80 TGFBR1 (0.50) TGFBR1CCR1CCR8CYP2A6GRM5
SCHEMBL3422361 0.78 CCR1 (0.75) TGFBR1CCR1CCR8ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed