SCHEMBL13680477

SCHEMBL13680477

Cc1cccc(-c2ccc(OC(F)(F)F)nc2)n1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.46
CCR1 P32246 1/20 0.43
CCR8 P51685 1/20 0.43
SCN9A Q15858 3/20 0.41
SCN10A Q9Y5Y9 1/20 0.39
BRS3 P32247 1/20 0.39
TGFBR1 P36897 6/20 0.38
GRM5 P41594 1/20 0.38
METAP2 P50579 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
DGAT1 O75907 1/20 0.36
SCN5A Q14524 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30146649 0.81 CYP2A6 (0.51) CYP2A6CCR1CCR8TGFBR1CYP1A2
SCHEMBL13680484 0.81 CYP2A6 (0.51) CYP2A6CCR1CCR8TGFBR1CYP1A2
SCHEMBL12269975 0.79 CYP19A1 (0.50) CYP2A6CCR1CCR8SCN9ABRS3
SCHEMBL10203331 0.78 SCN10A (0.53) CYP2A6CCR1CCR8SCN10ATGFBR1
SCHEMBL13680557 0.77 TRPV3 (0.51) CYP2A6CCR1CCR8SCN9ATGFBR1
SCHEMBL30146674 0.76 CYP2A6 (0.65) CYP2A6CCR1CCR8TGFBR1GRM5
SCHEMBL3421947 0.76 CYP2A6 (0.65) CYP2A6CCR1CCR8TGFBR1GRM5
SCHEMBL13680845 0.75 SCN9A (0.41) SCN9ACYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL13680445 0.75 HSD17B1 (0.46) SCN10A
SCHEMBL13680479 0.74 CYP2A6 (0.54) CYP2A6CCR1CCR8TGFBR1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed