SCHEMBL13680482

SCHEMBL13680482

Cc1csc(-c2ccc(C(N)=O)cc2)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 2/20 0.51
PIM1 P11309 1/20 0.49
PIM3 Q86V86 1/20 0.49
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PPARA Q07869 2/20 0.46
NPC1 O15118 5/20 0.45
RAB9A P51151 5/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
KDM4E B2RXH2 3/20 0.45
MAPT P10636 2/20 0.45
CYP2E1 P05181 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2A6 P11509 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2B6 P20813 1/20 0.45
AOC3 Q16853 2/20 0.45
GAA P10253 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680487 0.85 ALDH1A1 (0.49) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL13680478 0.85 KDM4E (0.62) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL13680733 0.83 CYP2E1 (0.45) TGFBR1ALDH1A1PPARANPC1RAB9A
SCHEMBL13681289 0.83 PPARA (0.46) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL8198560 0.82 CYP3A4 (0.60) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL31341074 0.81 MKNK1 (0.50) PIM1PIM3ALDH1A1MEN1KMT2A
SCHEMBL13680524 0.81 MAPT (0.58) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL13680527 0.81 RAB9A (0.66) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL13680528 0.81 ALDH1A1 (0.45) ALDH1A1MEN1KMT2APPARANPC1
SCHEMBL7905176 0.80 CYP3A4 (0.58) ALDH1A1MEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed