SCHEMBL13680478

SCHEMBL13680478

Cc1csc(-c2ccc(C(=O)O)cc2)n1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.62
RAB9A P51151 8/20 0.62
NPC1 O15118 7/20 0.62
SMN1; SMN2 Q16637 6/20 0.62
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
ALDH1A1 P00352 4/20 0.58
GAA P10253 2/20 0.56
POLB P06746 1/20 0.55
HTT P42858 1/20 0.55
RARA P10276 2/20 0.51
RARB P10826 2/20 0.51
RARG P13631 2/20 0.51
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
PPARA Q07869 1/20 0.50
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680487 0.86 ALDH1A1 (0.49) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL7399253 0.85 EIF4E (0.52) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL13680482 0.85 TGFBR1 (0.51) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL8198560 0.83 CYP3A4 (0.60) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL13680524 0.82 MAPT (0.58) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL13680527 0.82 RAB9A (0.66) RAB9ANPC1SMN1; SMN2MEN1KMT2A
SCHEMBL13680528 0.82 ALDH1A1 (0.45) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL7905176 0.81 CYP3A4 (0.58) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL13681289 0.81 PPARA (0.46) KDM4ERAB9ANPC1SMN1; SMN2MEN1
SCHEMBL3741835 0.81 KDM4E (0.49) KDM4ERAB9ANPC1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115286592-A GLUT1 inhibitor, virtual screening method and application 武汉工程大学 2022-11-04 CN disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed