SCHEMBL13680487

SCHEMBL13680487

CC(=O)c1ccc(-c2nc(C)cs2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
PPARA Q07869 2/20 0.47
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
CYP2E1 P05181 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2A6 P11509 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2B6 P20813 1/20 0.46
POLB P06746 1/20 0.45
EIF4E P06730 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B1 P14061 1/20 0.44
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43
PIK3CB P42338 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680478 0.86 KDM4E (0.62) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL13680482 0.85 TGFBR1 (0.51) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL8198560 0.83 CYP3A4 (0.60) ALDH1A1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL13680731 0.83 CYP3A4 (0.46) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL13680524 0.82 MAPT (0.58) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL13680528 0.82 ALDH1A1 (0.45) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL13680527 0.82 RAB9A (0.66) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL7905176 0.81 CYP3A4 (0.58) ALDH1A1NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL13681289 0.81 PPARA (0.46) ALDH1A1PPARANPC1RAB9ASMN1; SMN2
SCHEMBL13043927 0.81 EIF4E (0.52) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed