SCHEMBL13680564

SCHEMBL13680564

Cc1cccc(-c2ccc3c(c2)CC(=O)O3)n1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.41
CCR1 P32246 1/20 0.41
CCR8 P51685 1/20 0.41
MAOA P21397 4/20 0.39
MAOB P27338 4/20 0.39
TGFBR1 P36897 6/20 0.37
MAPK14 Q16539 2/20 0.37
RIPK2 O43353 1/20 0.37
ACVR1B P36896 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2615988 0.75 RAB9A (0.56) CCR1CCR8TGFBR1MAPK14RIPK2
SCHEMBL13680623 0.74 NPC1 (0.41) CYP2A6TGFBR1
SCHEMBL4761923 0.74 ALDH1A1 (0.48) MAOAMAOBTGFBR1
SCHEMBL13680566 0.73 PRF1 (0.52)
SCHEMBL27439272 0.73 MAOA (0.40) MAOAMAOB
SCHEMBL13680572 0.72 GRIA1 (0.62) TGFBR1
SCHEMBL15984797 0.72 NPC1 (0.57) CCR1CCR8TGFBR1MAPK14RIPK2
SCHEMBL15849494 0.72 TGFBR1 (0.62) TGFBR1MAPK14RIPK2ACVR1BTDP1
SCHEMBL13680668 0.71 CYP1A2 (0.50) CYP2A6CCR1CCR8TGFBR1
SCHEMBL31432603 0.70 CA12 (0.48) MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed