SCHEMBL13680588

SCHEMBL13680588

Cc1cccc(-c2ccc3nc[nH]c3c2)n1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 4/20 0.60
CYP2D6 P10635 1/20 0.60
TGFBR2 P37173 1/20 0.60
MAP3K20 Q9NYL2 1/20 0.60
QPCT Q16769 7/20 0.50
QPCTL Q9NXS2 5/20 0.50
BRD4 O60885 1/20 0.50
CREBBP Q92793 1/20 0.50
KDM4E B2RXH2 2/20 0.49
NPC1 O15118 1/20 0.49
ALDH1A1 P00352 1/20 0.49
TP53 P04637 1/20 0.49
HPGD P15428 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CCR1 P32246 1/20 0.46
CCR8 P51685 1/20 0.46
MMP12 P39900 1/20 0.45
PRKCI P41743 1/20 0.45
PSMD11 O00231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15640140 0.85 TGFBR1 (0.55) TGFBR1CYP2D6TGFBR2MAP3K20QPCT
SCHEMBL6760983 0.81 TGFBR1 (0.71) TGFBR1CYP2D6TGFBR2MAP3K20KDM4E
SCHEMBL13680559 0.78 RAB9A (0.56) TGFBR1KDM4ENPC1ALDH1A1HPGD
SCHEMBL13680531 0.78 QPCT (0.60) QPCTQPCTLBRD4CREBBPKDM4E
SCHEMBL8634290 0.77 QPCT (0.68) QPCTQPCTLBRD4CREBBPKDM4E
SCHEMBL11235922 0.76 QPCT (0.58) TGFBR1TGFBR2QPCTQPCTLBRD4
SCHEMBL25942078 0.76 TGFBR1 (0.73) TGFBR1CYP2D6TGFBR2MAP3K20QPCT
SCHEMBL15551561 0.74 QPCT (0.65) QPCTQPCTLBRD4CREBBPKDM4E
SCHEMBL21364016 0.74 TGFBR1 (0.55) TGFBR1CYP2D6TGFBR2MAP3K20
SCHEMBL22418756 0.73 QPCT (0.64) QPCTQPCTLKDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed