SCHEMBL13680684

SCHEMBL13680684

Cc1cccc(-c2cnc(N3CCCC3)nc2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.46
CCR1 P32246 1/20 0.46
CCR8 P51685 1/20 0.46
CYP2A6 P11509 1/20 0.45
CNR2 P34972 2/20 0.41
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
AOC3 Q16853 3/20 0.39
SIGMAR1 Q99720 1/20 0.39
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
THRB P10828 1/20 0.39
TGFBR1 P36897 1/20 0.39
DHFR P00374 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680682 0.87 PIK3CA (0.52) CNR2ALDH1A1AOC3POLB
SCHEMBL13680685 0.87 KCNH2 (0.49) CCR1CCR8CYP2A6ALDH1A1
SCHEMBL19626523 0.78 CCR1 (0.48) HRH3CCR1CCR8CYP2A6NPC1
SCHEMBL13680679 0.76 CCR1 (0.60) CCR1CCR8CYP2A6RAB9ATGFBR1
SCHEMBL16122790 0.76 CNR2 (0.65) HRH3CCR1CCR8CYP2A6CNR2
SCHEMBL12269941 0.75 CAMK2D (0.47) CCR1CCR8CYP2A6DHFR
SCHEMBL13680656 0.73 AOC3 (0.51) NPC1ALDH1A1RAB9AAOC3SIGMAR1
SCHEMBL13680673 0.73 CCR1 (0.56) CCR1CCR8CYP2A6TGFBR1METAP2
SCHEMBL8241132 0.72 ALDH1A1 (0.48) NPC1ALDH1A1RAB9APOLBSMN1; SMN2
SCHEMBL13606215 0.72 AOC3 (0.52) CNR2NPC1ALDH1A1RAB9AAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed