SCHEMBL13680685

SCHEMBL13680685

Cc1cccc(-c2cnc(N3CCNCC3)nc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.49
CACNA1C Q13936 1/20 0.49
ASIC3 Q9UHC3 1/20 0.49
MAPT P10636 1/20 0.49
TAAR1 Q96RJ0 1/20 0.47
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 1/20 0.46
PIM1 P11309 4/20 0.43
CYP2A6 P11509 1/20 0.42
CCR1 P32246 1/20 0.42
CCR8 P51685 1/20 0.42
PIM3 Q86V86 3/20 0.41
PIM2 Q9P1W9 3/20 0.41
KARS1 Q15046 1/20 0.41
CYP1A2 P05177 3/20 0.41
HPGD P15428 3/20 0.41
CASP1 P29466 3/20 0.41
CASP7 P55210 3/20 0.41
HSD17B10 Q99714 3/20 0.41
CYP3A4 P08684 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680684 0.87 HRH3 (0.46) ALDH1A1CYP2A6CCR1CCR8
SCHEMBL13680682 0.83 PIK3CA (0.52) KCNH2MAPTALDH1A1
Hydrochloric Acid SCHEMBL22371670 0.78 MAPKAPK2 (0.46) MAPTTAAR1ALDH1A1KDM4EPIM1
SCHEMBL30156515 0.77 TGFBR1 (0.40) KCNH2CACNA1CASIC3PIM1PIM3
SCHEMBL25085386 0.77 TGFBR1 (0.40) KCNH2CACNA1CASIC3PIM1PIM3
SCHEMBL4582036 0.75 ADRB1 (0.54) TAAR1ALDH1A1KDM4ECYP1A2HPGD
SCHEMBL4582837 0.74 HTR1A (0.54) KCNH2CACNA1CASIC3MAPTTAAR1
SCHEMBL9400977 0.73 TAAR1 (0.64) TAAR1ALDH1A1KDM4ECYP1A2HPGD
SCHEMBL7991455 0.72 ALDH1A1 (0.59) TAAR1ALDH1A1KDM4ECYP1A2HPGD
SCHEMBL13680679 0.72 CCR1 (0.60) CYP2A6CCR1CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed