SCHEMBL13680544

SCHEMBL13680544

COC(=O)Nc1cccc(-c2cccc(C)n2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 10/20 0.51
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
MAPT P10636 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
FAAH O00519 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
MAPK1 P28482 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
FYN P06241 2/20 0.46
FGFR3 P22607 1/20 0.45
KDR P35968 1/20 0.45
CNR2 P34972 1/20 0.45
CYP2A6 P11509 1/20 0.45
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12318239 0.85 NPC1 (0.62) CNR1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL13537053 0.85 SMN1; SMN2 (0.49) NPC1RAB9AMAPTSMN1; SMN2NFKB1
SCHEMBL11653085 0.81 MGLL (0.58) CNR1SMN1; SMN2FAAHALDH1A1CYP3A4
SCHEMBL13680584 0.78 GABRG2 (0.53) NPC1RAB9AMAPK1CYP2A6TP53
SCHEMBL13680515 0.77 FAAH (0.66) CNR1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL13680686 0.77 CYP2A6 (0.45) NPC1RAB9AMAPTSMN1; SMN2MEN1
SCHEMBL2094875 0.77 MGLL (0.68) CNR1FAAHMEN1KMT2A
SCHEMBL14636653 0.76 CNR1 (0.47) CNR1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL716889 0.76 MAPK1 (0.62) NPC1RAB9AMAPTSMN1; SMN2FAAH
SCHEMBL13680552 0.75 CYP2A6 (0.53) FYNKDRCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed