SCHEMBL13680709

SCHEMBL13680709

Cc1ccc(-c2cnc(N(C)C)nc2)o1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.37
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 3/20 0.37
LMNA P02545 3/20 0.37
NPC1 O15118 3/20 0.37
HPGD P15428 3/20 0.37
RAB9A P51151 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37
HSD17B10 Q99714 2/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
ALOX15 P16050 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PTGS1 P23219 1/20 0.35
PTGS2 P35354 1/20 0.35
APP P05067 2/20 0.35
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
GSK3B P49841 2/20 0.33
AOC3 Q16853 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680715 0.80 TDP1 (0.42) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680505 0.79 APP (0.49) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680711 0.77 ALDH1A1 (0.39) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680718 0.77 ALDH1A1 (0.39) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680518 0.74 MAPT (0.41) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680700 0.74 MAP4K4 (0.41) GRM5ALDH1A1KDM4ELMNANPC1
SCHEMBL13680720 0.74 GSK3B (0.38) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680469 0.73 NPC1 (0.42) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13681360 0.73 ALDH1A1 (0.40) ALDH1A1KDM4ELMNANPC1HPGD
SCHEMBL13680704 0.73 SMN1; SMN2 (0.53) ALDH1A1KDM4ELMNANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed