SCHEMBL13709449

SCHEMBL13709449

N=C1CC(COCC(=O)O)N(C(=O)c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 2/20 0.39
OXTR P30559 2/20 0.39
AVPR1A P37288 1/20 0.39
HPGD P15428 2/20 0.38
MAPK1 P28482 1/20 0.38
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
POLB P06746 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
SLC6A7 Q99884 1/20 0.35
TSHR P16473 2/20 0.35
FASN P49327 1/20 0.35
ABCB1 P08183 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8343791 0.87 OXTR (0.37) NR1D1OXTRAVPR1AHPGDMAPK1
SCHEMBL8343604 0.86 OXTR (0.44) NR1D1OXTRAVPR1AHPGDMAPK1
SCHEMBL8342472 0.83 LMNA (0.42) NR1D1OXTRAVPR1AHPGDMAPK1
SCHEMBL8342892 0.83 OXTR (0.50) OXTRAVPR1AHPGDMAPK1MEN1
SCHEMBL8341758 0.82 FFAR4 (0.37) HPGDMAPK1SMN1; SMN2LMNA
SCHEMBL8341237 0.82 HPGD (0.42) OXTRAVPR1AHPGDMAPK1MEN1
SCHEMBL13709473 0.81 ACHE (0.46) HPGDMEN1KMT2APOLB
SCHEMBL4418459 0.81 OXTR (0.61) NR1D1OXTRAVPR1AHPGDMAPK1
SCHEMBL8338121 0.81 HPGD (0.41) OXTRAVPR1AHPGDMAPK1MEN1
SCHEMBL8344306 0.77 OXTR (0.41) OXTRAVPR1AHPGDMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532109-B1 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS MERCK SERONO SA (CH) 2009-09-09 EP disclosed