SCHEMBL8341237

SCHEMBL8341237

N=C1CC(CN)N(C(=O)c2ccc(-c3ccccc3)cc2)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
POLB P06746 3/20 0.40
OXTR P30559 2/20 0.39
AVPR1A P37288 1/20 0.39
SLC6A7 Q99884 1/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 2/20 0.39
FASN P49327 1/20 0.39
ABCB1 P08183 1/20 0.39
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
NR2F2 P24468 1/20 0.37
RAB9A P51151 1/20 0.37
BDKRB2 P30411 1/20 0.37
SMYD3 Q9H7B4 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8342892 0.88 OXTR (0.50) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL8338121 0.86 HPGD (0.41) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL4418365 0.85 HPGD (0.43) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL4418361 0.85 HPGD (0.43) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL8343604 0.84 OXTR (0.44) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL8344306 0.82 OXTR (0.41) HPGDMAPK1SMN1; SMN2POLBOXTR
SCHEMBL13709449 0.82 NR1D1 (0.39) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL8341197 0.82 HPGD (0.47) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL8342472 0.81 LMNA (0.42) HPGDMAPK1SMN1; SMN2MEN1KMT2A
SCHEMBL13709427 0.81 MMP2 (0.43) HPGDMAPK1SMN1; SMN2POLBOXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1532109-B1 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS MERCK SERONO SA (CH) 2009-09-09 EP disclosed
WO-2004005249-A1 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-01-15 WO disclosed