SCHEMBL1374248

SCHEMBL1374248

O=C(O)CCC(NC(=O)NC(CS)C(=O)O)C(=O)O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 8/20 1.00
NAALAD2 Q9Y3Q0 7/20 0.81
RIMKLA Q8IXN7 1/20 0.81
KDM4E B2RXH2 1/20 0.52
MAPT P10636 1/20 0.52
THRB P10828 1/20 0.52
ALOX15 P16050 1/20 0.52
NFKB1 P19838 1/20 0.52
PTGS2 P35354 1/20 0.52
THPO P40225 1/20 0.52
RECQL P46063 1/20 0.52
BLM P54132 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21321511 1.00 FOLH1 (1.00) FOLH1NAALAD2RIMKLAKDM4EMAPT
SCHEMBL19209754 1.00 FOLH1 (1.00) FOLH1NAALAD2RIMKLAKDM4EMAPT
SCHEMBL11936653 1.00 FOLH1 (1.00) FOLH1NAALAD2RIMKLAKDM4EMAPT
SCHEMBL12145776 0.90 FOLH1 (1.00) FOLH1NAALAD2RIMKLA
SCHEMBL18161468 0.90 FOLH1 (1.00) FOLH1NAALAD2RIMKLA
SCHEMBL1377049 0.90 FOLH1 (1.00) FOLH1NAALAD2RIMKLA
SCHEMBL14102890 0.90 FOLH1 (1.00) FOLH1NAALAD2RIMKLA
SCHEMBL14102870 0.90 FOLH1 (1.00) FOLH1NAALAD2RIMKLA
SCHEMBL19259307 0.89 FOLH1 (0.81) FOLH1NAALAD2RIMKLA
SCHEMBL18636844 0.89 FOLH1 (0.81) FOLH1NAALAD2RIMKLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 95 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180338910-A1 INTRANASAL ADMINISTRATION OF GLUTAMATE CARBOXYPEPTIDASE (GCP-II) INHIBITORS THE JOHNS HOPKINS UNIVERSITY (US) 2018-11-29 US claimed
US-12496292-B2 PSMA binding ligand-linker conjugates and methods for using PURDUE RESEARCH FOUNDATION (US) 2025-12-16 US disclosed
EP-4648799-A1 LIGAND-DRUG CONJUGATES Sun Pharma Advanced Research Company Ltd (IN) 2025-11-19 EP disclosed
US-20250127939-A1 COMPOUNDS FOR POSITRON EMISSION TOMOGRAPHY PURDUE RESEARCH FOUNDATION 2025-04-24 US disclosed
EP-4541378-A2 COMPOUNDS FOR POSITRON EMISSION TOMOGRAPHY Endocyte, Inc. (US) 2025-04-23 EP disclosed
US-20250108039-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION 2025-04-03 US disclosed
US-12252534-B2 Humanized anti-CD3 antibodies, conjugates and uses thereof THE SCRIPPS RESEARCH INSTITUTE (US) 2025-03-18 US disclosed
EP-3838298-B1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2025-02-26 EP disclosed
EP-3777898-B1 COMPOUNDS FOR POSITRON EMISSION TOMOGRAPHY ENDOCYTE INC (US) 2025-01-01 EP disclosed
US-12178892-B2 Compounds for positron emission tomography PURDUE RESEARCH FOUNDATION (US) 2024-12-31 US disclosed
US-20140073763-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2014-03-13 US disclosed
US-20130011362-A1 TARGETING MONOMERS AND POLYMERS HAVING TARGETING BLOCKS PHASERX, INC. (US) 2013-01-10 US disclosed
US-20120276007-A1 IMAGING AGENTS AND METHODS OF IMAGING NAALADASE OR PSMA GEORGETOWN UNIVERSITY (US) 2012-11-01 US disclosed
US-20110288152-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2011-11-24 US disclosed
US-20100324008-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2010-12-23 US disclosed
EP-2187965-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2010-05-26 EP disclosed
WO-2010045598-A2 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2010-04-22 WO disclosed
WO-2009026177-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING PURDUE RESEARCH FOUNDATION (US) 2009-02-26 WO disclosed
US-20080311037-A1 Compounds which bind PSMA and uses thereof NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2008-12-18 US disclosed
US-20080311037-A1 Compounds which bind PSMA and uses thereof NATIONAL INSTITUTES OF HEALTH - DIRECTOR DEITR 2008-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130011362-A1 TARGETING MONOMERS AND POLYMERS HAVING TARGETING BLOCKS FOLR1, FOLR2, DHFR FOLH1 14/4885NAALAD2 3927/4885RIMKLA 675/4885
US-20110288152-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING FOLH1, KLK3, PSMA1 FOLH1 1/4885NAALAD2 32/4885RIMKLA 801/4885
US-20250108039-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING FOLH1, KLK3, PSMA1 FOLH1 1/4885NAALAD2 49/4885RIMKLA 513/4885
US-20180338910-A1 INTRANASAL ADMINISTRATION OF GLUTAMATE CARBOXYPEPTIDASE (GCP-II) INHIBITORS ENPEP, DNPEP, FOLH1 FOLH1 3/4885NAALAD2 29/4885RIMKLA 121/4885
US-12496292-B2 PSMA binding ligand-linker conjugates and methods for using FOLH1, KLK3, PSMA1 FOLH1 1/4885NAALAD2 49/4885RIMKLA 513/4885
US-20080311037-A1 Compounds which bind PSMA and uses thereof FOLH1, PSMA1, BPHL FOLH1 1/4885NAALAD2 208/4885RIMKLA 1263/4885
US-20250127939-A1 COMPOUNDS FOR POSITRON EMISSION TOMOGRAPHY VHL, PC, NPC1 FOLH1 157/4885NAALAD2 659/4885RIMKLA 874/4885
US-12178892-B2 Compounds for positron emission tomography FOLH1, FOLR2, FOLR1 FOLH1 1/4885NAALAD2 67/4885RIMKLA 110/4885
US-12252534-B2 Humanized anti-CD3 antibodies, conjugates and uses thereof CD2, CD47, KLK3 FOLH1 43/4885NAALAD2 172/4885RIMKLA 2261/4885
US-20100324008-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING FOLH1, KLK3, PSMA1 FOLH1 1/4885NAALAD2 49/4885RIMKLA 513/4885
US-20140073763-A1 PSMA BINDING LIGAND-LINKER CONJUGATES AND METHODS FOR USING FOLH1, KLK3, PSMA1 FOLH1 1/4885NAALAD2 49/4885RIMKLA 513/4885
US-20120276007-A1 IMAGING AGENTS AND METHODS OF IMAGING NAALADASE OR PSMA FOLH1, DNPEP, NAALAD2 FOLH1 1/4885NAALAD2 3/4885RIMKLA 197/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.