SCHEMBL13748458

SCHEMBL13748458

Cc1cc(-n2cc3c(n2)CCN(CC(=O)N2CCN(C(C)C)CC2)C3)ccn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 9/20 0.44
KCNH2 Q12809 5/20 0.44
PDK2 Q15119 1/20 0.34
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
TSHR P16473 1/20 0.34
ENPP2 Q13822 1/20 0.34
TLR9 Q9NR96 1/20 0.34
TLR8 Q9NR97 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
CHRM4 P08173 1/20 0.33
PRMT5 O14744 1/20 0.33
WDR77 Q9BQA1 1/20 0.33
IDO1 P14902 1/20 0.33
S1PR1 P21453 1/20 0.33
CDK1 P06493 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13749141 0.90 SLC6A9 (0.43) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13748065 0.90 ALDH1A1 (0.42) SLC6A9KCNH2KMT2AKDM4EMEN1
SCHEMBL13749100 0.89 SLC6A9 (0.42) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13748398 0.89 KMT2A (0.35) KCNH2PDK2KMT2AKDM4EMEN1
SCHEMBL13748801 0.87 SLC6A9 (0.41) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13748459 0.87 SLC6A9 (0.44) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13748331 0.86 ALDH1A1 (0.47) SLC6A9KCNH2KMT2AMEN1ALDH1A1
SCHEMBL13748980 0.86 SLC6A9 (0.41) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13749140 0.86 SLC6A9 (0.41) SLC6A9KCNH2PDK2KMT2AKDM4E
SCHEMBL13749042 0.86 SLC6A9 (0.41) SLC6A9KCNH2PDK2KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100120-A2 PYRIDINYL-SUBSTITUTED PIPERAZINYL OXOETHYL TETRAHYDROPYRAZOLOPYRIDINES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed