SCHEMBL13763543

SCHEMBL13763543

CCc1ccc(NCCNC(C)=O)nc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 5/20 0.47
PDCD1 Q15116 2/20 0.43
CD274 Q9NZQ7 2/20 0.43
CYP1A2 P05177 5/20 0.43
CLK4 Q9HAZ1 3/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP3A4 P08684 3/20 0.43
HSD17B10 Q99714 3/20 0.43
ALOX15 P16050 2/20 0.43
MAPK1 P28482 1/20 0.43
DEGS1 O15121 1/20 0.43
KDM4E B2RXH2 1/20 0.41
F13A1 P00488 1/20 0.41
TDO2 P48775 1/20 0.41
ACACB O00763 2/20 0.41
TSHR P16473 2/20 0.40
CYP2C9 P11712 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1108653 0.81 RAB9A (0.53) HCAR3CYP1A2CLK4ALDH1A1CYP3A4
SCHEMBL7238262 0.80 HCAR3 (0.44) HCAR3CYP1A2CLK4ALDH1A1CYP3A4
SCHEMBL12693710 0.79 HCAR3 (0.45) HCAR3CLK4ALDH1A1DEGS1KDM4E
SCHEMBL2759546 0.79 PTK2 (0.59) HCAR3CYP1A2DEGS1KDM4E
SCHEMBL12327198 0.79 HCAR3 (0.56) HCAR3ALDH1A1MAPK1DEGS1KDM4E
SCHEMBL25056983 0.77 PRKAB2 (0.60) CYP1A2CLK4ALDH1A1CYP3A4HSD17B10
SCHEMBL7233175 0.75 GAA (0.65) CYP1A2ALDH1A1
SCHEMBL14416655 0.75 HCAR3 (0.53) HCAR3CYP1A2ALDH1A1MAPK1DEGS1
SCHEMBL11466907 0.74 DEGS1 (0.56) HCAR3HSD17B10DEGS1
SCHEMBL8145501 0.73 CYP1A2 (0.56) CYP1A2CLK4ALDH1A1CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579348-B2 Derivatives of 8-substituted xanthines PGXHEALTH, LLC (US) 2009-08-25 US disclosed