SCHEMBL7238262

SCHEMBL7238262

CC(=O)NCCNc1ccc(N)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 5/20 0.44
CYP1A2 P05177 6/20 0.44
CYP3A4 P08684 5/20 0.44
HSD17B10 Q99714 5/20 0.44
ALDH1A1 P00352 4/20 0.44
ALOX15 P16050 4/20 0.44
CLK4 Q9HAZ1 3/20 0.44
MAPK1 P28482 1/20 0.44
TDO2 P48775 1/20 0.42
POLB P06746 1/20 0.42
TSHR P16473 2/20 0.41
CYP2C9 P11712 1/20 0.41
PTGS1 P23219 1/20 0.40
FTO Q9C0B1 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM5B Q9UGL1 1/20 0.40
KDM2A Q9Y2K7 1/20 0.40
KDM3A Q9Y4C1 1/20 0.40
CA12 O43570 1/20 0.40
CA4 P22748 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29395019 0.87 POLB (0.43) HCAR3POLBPTGS1FTOKDM4C
SCHEMBL29170287 0.86 POLB (0.43) HCAR3POLBPTGS1FTOKDM4C
SCHEMBL3943928 0.86 HCAR3 (0.45) HCAR3ALDH1A1POLBPTGS1FTO
SCHEMBL29394423 0.84 POLB (0.42) HCAR3ALDH1A1POLBTSHRPTGS1
SCHEMBL30639140 0.83 HRH4 (0.45) HCAR3ALDH1A1POLBPTGS1FTO
SCHEMBL11252790 0.83 HRH4 (0.45) HCAR3ALDH1A1POLBPTGS1FTO
SCHEMBL1108653 0.83 RAB9A (0.53) HCAR3CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL13947394 0.80 LMNA (0.52) HCAR3POLBTSHRPTGS1LMNA
SCHEMBL13763543 0.80 HCAR3 (0.47) HCAR3CYP1A2CYP3A4HSD17B10ALDH1A1
SCHEMBL13685154 0.79 PTGS1 (0.43) HCAR3PTGS1FTOKDM4CKDM5B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6599908-B1 Potent and selective inhibitors of the protein tyrosine kinases p56lck and p59fyn CELLTECH R & D LIMITED (GB) 2003-07-29 US disclosed
US-6057329-A Fused polycyclic 2-aminopyrimidine derivatives CELLTECH THERAPEUTICS LIMITED (GB) 2000-05-02 US disclosed