SCHEMBL13767982

SCHEMBL13767982

COC(=O)c1cncc(N2CC3CC(C2)N(C(=O)OC(C)(C)C)C3)c1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 8/20 0.40
CHRNA3 P32297 8/20 0.40
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
ATM Q13315 1/20 0.37
UCHL1 P09936 1/20 0.36
USP30 Q70CQ3 1/20 0.36
HDAC1 Q13547 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
HSD11B1 P28845 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13768041 0.84 HSD11B1 (0.38) HDAC1HSD11B1NR1H2NR1H3
SCHEMBL13768188 0.84 HTT (0.39) CHRNB4CHRNA3CHRNB2CHRNA4HDAC1
SCHEMBL4119940 0.84 HSD11B1 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4UCHL1
SCHEMBL13768190 0.82 AR (0.43) CHRNB4CHRNA3CHRNB2CHRNA4NR1H2
SCHEMBL13768179 0.81 CHRNB4 (0.48) CHRNB4CHRNA3USP30HDAC1HSD11B1
SCHEMBL13768039 0.80 CHRNB2 (0.39) CHRNB4CHRNA3CHRNB2CHRNA4HDAC1
SCHEMBL13768040 0.79 HDAC1 (0.38) CHRNB4CHRNA3HDAC1HSD11B1NR1H2
SCHEMBL13768184 0.77 GPR119 (0.35) CHRNB4CHRNA3HDAC1HSD11B1NR1H2
SCHEMBL23572659 0.76 GPR119 (0.48) ATMNR1H2
SCHEMBL25614203 0.75 CHRNB4 (0.50) CHRNB4CHRNA3CHRNB2CHRNA4ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081246-A2 BICYCLIC DIAMINES AS NICOTINIC RECEPTOR AGONISTS PFIZER INC. (US) 2009-07-02 WO disclosed