SCHEMBL13801192

SCHEMBL13801192

Cc1cccc(-n2nnnc2C(F)(F)F)n1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.40
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR3A P46098 1/20 0.38
HTR3D Q70Z44 1/20 0.38
HTR3C Q8WXA8 1/20 0.38
RECQL P46063 1/20 0.38
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.36
CACNA1B Q00975 2/20 0.36
APBA1 Q02410 2/20 0.36
HSP90AA1 P07900 1/20 0.36
IRAK4 Q9NWZ3 7/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CCR6 P51684 1/20 0.35
NOTUM Q6P988 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12435278 0.78 HTR3E (0.43) P2RX7HTR3EHTR3BHTR3AHTR3D
SCHEMBL25620027 0.73 MAP3K5 (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL5551503 0.70 ALDH1A1 (0.70) ALDH1A1MAPTHPGDHTTCACNA1B
SCHEMBL7916517 0.70 TACR1 (0.36) ALDH1A1MAPTHPGD
SCHEMBL4408113 0.69 ALDH1A1 (0.68) ALDH1A1MAPTHPGDHTTCACNA1B
SCHEMBL5551521 0.69 ALDH1A1 (0.46) ALDH1A1MAPTHPGDHTTCACNA1B
SCHEMBL6923107 0.67 TACR1 (0.36) ALDH1A1MAPTHPGD
SCHEMBL4204766 0.67 ALDH1A1 (0.58) ALDH1A1MAPTHPGDHTTCACNA1B
SCHEMBL4210628 0.65 ALDH1A1 (0.43) ALDH1A1MAPTHPGDHTTCACNA1B
SCHEMBL6541068 0.65 NOTUM (0.46) ALDH1A1MAPTHPGDHTTCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE48334-E1 Nitrogen-containing heterocyclic compound and use of same TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2020-12-01 US disclosed
US-8470816-B2 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-25 US disclosed
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED 2009-06-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090156572-A1 Nitrogen-containing heterocyclic compound and use thereof NTSR2, NTSR1, HNMT P2RX7 941/4885HTR3E 215/4885HTR3B 96/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.